SCHEMBL11748801

SCHEMBL11748801

Clc1cccc(-c2nc(Cl)sc2-c2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.53
ADORA2A P29274 4/20 0.53
KDM1A O60341 1/20 0.51
PTGS1 P23219 1/20 0.48
PTGS2 P35354 1/20 0.48
NPC1 O15118 1/20 0.47
TP53 P04637 1/20 0.47
TSHR P16473 1/20 0.47
NFKB1 P19838 1/20 0.47
RAB9A P51151 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
IDO1 P14902 1/20 0.46
ALDH1A1 P00352 3/20 0.46
MAPT P10636 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
ADORA2B P29275 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11749855 0.93 ADORA1 (0.53) ADORA1ADORA2AKDM1APTGS1PTGS2
SCHEMBL11754235 0.93 ADORA2A (0.47) ADORA1ADORA2AKDM1APTGS1PTGS2
SCHEMBL11753179 0.86 ALDH1A1 (0.60) KDM1APTGS1PTGS2SMN1; SMN2ALDH1A1
SCHEMBL11751671 0.84 LMNA (0.54) ADORA1ADORA2AKDM1APTGS2SMN1; SMN2
SCHEMBL11753711 0.84 RORB (0.47) KDM1ANPC1TP53TSHRRAB9A
SCHEMBL11755296 0.83 KDM4E (0.55) KDM1APTGS1PTGS2NPC1RAB9A
SCHEMBL11752931 0.83 KDM4E (0.55) KDM1APTGS1PTGS2NPC1RAB9A
SCHEMBL11753624 0.81 ADORA2A (0.50) ADORA1ADORA2ANPC1TP53NFKB1
SCHEMBL11751969 0.79 LMNA (0.48) NPC1TSHRRAB9ARELASMN1; SMN2
SCHEMBL11751150 0.79 ADORA1 (0.58) ADORA1ADORA2ANPC1TP53NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4051250-A OXAZOLE, THIAZOLE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-27 US disclosed
US-3933840-A ANTIPHLOGISTIC MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-01-20 US disclosed