SCHEMBL11775697

SCHEMBL11775697

Nc1cccc(C(=O)CC(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PBRM1 Q86U86 1/20 0.50
PTGS1 P23219 5/20 0.48
ACHE P22303 1/20 0.44
NPC1 O15118 1/20 0.44
MITF O75030 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
F2 P00734 1/20 0.43
PLG P00747 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
ELANE P08246 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7913955 0.83 ACHE (0.56) PBRM1PTGS1ACHENPC1MITF
SCHEMBL6154661 0.82 PBRM1 (0.50) PBRM1PTGS1ACHENPC1MITF
SCHEMBL3260498 0.81 PBRM1 (0.49) PBRM1PTGS1ACHENPC1MITF
SCHEMBL11768399 0.80 CA12 (0.52) ACHENPC1LMNAKDM4EALDH1A1
SCHEMBL28359889 0.79 PBRM1 (0.59) PBRM1PTGS1NPC1MITFLMNA
SCHEMBL23217892 0.79 PARP1 (0.52) ACHENPC1ALDH1A1SMN1; SMN2RECQL
SCHEMBL633209 0.77 PBRM1 (0.57) PBRM1PTGS1NPC1MITFLMNA
SCHEMBL3373649 0.77 PBRM1 (0.57) PBRM1PTGS1NPC1MITFLMNA
SCHEMBL3801679 0.77 ANPEP (0.43) ACHECES2
SCHEMBL70367 0.77 CES1 (0.56) NPC1LMNAPOLBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3940407-A β-Adrenergic blocking agents in the 1,2,3-thiadiazole series SYNTEX (U.S.A.) INC. (US) 1976-02-24 US disclosed