SCHEMBL11778917

SCHEMBL11778917

COc1ccc2cc(N(C(=O)CO)C(C)C)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.50
AKR1C3 P42330 7/20 0.46
AKR1C2 P52895 7/20 0.46
PTGS1 P23219 4/20 0.46
PTGS2 P35354 3/20 0.46
TSHR P16473 2/20 0.46
CYP1A2 P05177 2/20 0.46
CDC42 P60953 1/20 0.46
RAC1 P63000 1/20 0.46
SLC22A6 Q4U2R8 1/20 0.46
ALOX5 P09917 2/20 0.44
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
CYP2C9 P11712 1/20 0.43
KDM4E B2RXH2 2/20 0.43
AKR1C1 Q04828 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10537588 0.86 TRPM8 (0.49) TSHRLMNAMAPTNPC1TP53
SCHEMBL11782640 0.81 AKR1C3 (0.46) ABCB11AKR1C3AKR1C2PTGS1PTGS2
SCHEMBL11778122 0.78 ABCB11 (0.43) ABCB11AKR1C3AKR1C2PTGS1PTGS2
SCHEMBL9877199 0.76 NQO1 (0.45) TSHRLMNAMAPTKDM4ETDP1
SCHEMBL10982814 0.74 ALOX5 (0.41) AKR1C3AKR1C2PTGS1PTGS2TSHR
SCHEMBL25316112 0.73 ALDH1A1 (0.66) LMNAMAPTKDM4ETDP1NPC1
SCHEMBL4868746 0.73 TRPM8 (0.48) TSHRALOX5LMNAMAPTNPC1
SCHEMBL4869949 0.73 GSK3B (0.49) TSHRLMNAMAPTNPC1TP53
Methane SCHEMBL11294998 0.72 ABCB11 (0.42) ABCB11AKR1C3AKR1C2PTGS1PTGS2
SCHEMBL8428661 0.71 MTNR1A (0.46) LMNATP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3931269-A ANTIINFLAMMATORY WILLIAM H. RORER, INC. (US) 1976-01-06 US disclosed