SCHEMBL11903517

SCHEMBL11903517

COc1cc(-c2nc3cc(OC(F)(F)F)ccc3[nH]2)ccc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RUNX1 Q01196 2/20 0.52
TRPV1 Q8NER1 1/20 0.51
CYP1A1 P04798 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP1B1 Q16678 1/20 0.50
NOX1 Q9Y5S8 2/20 0.49
PARP1 P09874 1/20 0.47
AMY1A P0DUB6 3/20 0.45
CHEK1 O14757 2/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
BACE1 P56817 1/20 0.44
ALOX5 P09917 1/20 0.44
EPHX2 P34913 1/20 0.44
FYN P06241 1/20 0.43
SMPD3 Q9NY59 2/20 0.43
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903521 0.91 RUNX1 (0.63) RUNX1TRPV1CYP1A1CYP1A2CYP1B1
SCHEMBL11903647 0.84 TRPV1 (0.62) RUNX1TRPV1PARP1KDM4EALDH1A1
SCHEMBL7396876 0.81 ALOX5 (0.62) CYP1A1CYP1A2CYP1B1NOX1PARP1
SCHEMBL11903487 0.80 CYP1A2 (0.54) RUNX1TRPV1CYP1A2PARP1KDM4E
SCHEMBL7395692 0.80 AMY1A (0.62) CYP1A1CYP1A2CYP1B1NOX1PARP1
SCHEMBL11903530 0.79 PDE4A (0.59) RUNX1TRPV1ALOX5EPHX2KDM4E
SCHEMBL11903494 0.79 TRPV1 (0.62) RUNX1TRPV1ACHEKDM4EALDH1A1
SCHEMBL15456540 0.78 CYP1A1 (0.69) CYP1A1CYP1A2CYP1B1NOX1PARP1
SCHEMBL11903464 0.78 TRPV1 (0.60) RUNX1TRPV1BACE1KDM4EALDH1A1
SCHEMBL11903505 0.78 RUNX1 (0.57) RUNX1TRPV1CYP1A2AMY1AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed