SCHEMBL11903539

SCHEMBL11903539

Cc1csc(-c2nc3ccc(OC(F)(F)F)cc3[nH]2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.57
RUNX1 Q01196 7/20 0.54
CBFB Q13951 3/20 0.54
SCN10A Q9Y5Y9 1/20 0.46
P2RY6 Q15077 1/20 0.45
BACE1 P56817 1/20 0.45
CHEK2 O96017 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPBWR1 P48145 1/20 0.41
PDE10A Q9Y233 1/20 0.41
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903462 0.80 ALDH1A1 (0.60) TRPV1RUNX1CBFBSCN10AP2RY6
SCHEMBL11903498 0.80 TRPV1 (0.77) TRPV1RUNX1CBFBCHEK2NPBWR1
SCHEMBL10146526 0.76 TRPV1 (0.59) TRPV1RUNX1CBFBSCN10APDE10A
SCHEMBL11903652 0.74 TRPV1 (0.77) TRPV1RUNX1CBFBCHEK2NPBWR1
SCHEMBL11903481 0.74 TRPV1 (0.72) TRPV1RUNX1CBFBCHEK2CYP1A2
SCHEMBL902354 0.73 CBFB (0.64) TRPV1RUNX1CBFBSCN10AP2RY6
SCHEMBL11903468 0.73 TRPV1 (0.74) TRPV1RUNX1CBFBBACE1CHEK2
SCHEMBL11903447 0.72 TRPV1 (0.73) TRPV1RUNX1CBFBCHEK2CYP3A4
SCHEMBL11903519 0.72 TRPV1 (0.72) TRPV1RUNX1CBFBSCN10ACHEK2
SCHEMBL14475012 0.71 TRPV1 (0.54) TRPV1RUNX1CBFBSCN10AP2RY6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed