SCHEMBL11973236

SCHEMBL11973236

NC(=O)c1ccc2c(Cl)cc[c]c2n1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.38
LMNA P02545 1/20 0.38
GRM2 Q14416 6/20 0.35
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34
SIRT6 Q8N6T7 1/20 0.33
CHEK2 O96017 2/20 0.32
NNMT P40261 1/20 0.31
IKBKB O14920 1/20 0.31
PIM3 Q86V86 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4484391 0.81 GRM2 (0.35) PIM1LMNAGRM2NNMT
SCHEMBL3050408 0.78 PIM1 (0.33) PIM1GRM2NNMTIKBKB
SCHEMBL11973850 0.77 KMT2A (0.40) PIM1GRM2KMT2ASCN9A
SCHEMBL4473023 0.77 NNMT (0.41) PIM1GRM2SIRT6NNMTIKBKB
SCHEMBL16742949 0.72 LMNA (0.45) PIM1LMNAGRM2SIRT6CHEK2
SCHEMBL19329369 0.71 PIM1 (0.49) PIM1LMNAKMT2ANNMT
SCHEMBL5447337 0.70 GRM2 (0.35) PIM1LMNAGRM2NNMTIKBKB
SCHEMBL18343855 0.70 PIM1 (0.38) PIM1LMNAGRM2KMT2ASIRT6
SCHEMBL5447285 0.68 GRM2 (0.33) PIM1GRM2NNMTIKBKB
SCHEMBL3341422 0.68 GRM2 (0.41) PIM1GRM2IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675526-B1 NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS VIFOR (INTERNATIONAL) AG (CH) 2017-02-01 EP disclosed
US-9102688-B2 Sulfonaminoquinoline hepcidin antagonists VIFOR (INTERNATIONAL) AG (CH) 2015-08-11 US disclosed
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2014-12-11 US disclosed
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists VIFOR (INTERNATIONAL) AG (CH) 2012-08-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120214803-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists HAMP, SLC40A1, FTH1 PIM1 2312/4885LMNA 4127/4885GRM2 3667/4885
US-20140364424-A1 Novel Sulfonaminoquinoline Hepcidin Antagonists HAMP, SLC40A1, FTH1 PIM1 2312/4885LMNA 4127/4885GRM2 3667/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.