Norcodeine

Norcodeine

SCHEMBL120270

COc1ccc2c3c1O[C@H]1[C@@H](O)C=C[C@H]4[C@@H](C2)NCC[C@@]341

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MRGPRX2 Q96LB1 5/20 1.00
MAPT P10636 1/20 1.00
OPRM1 P35372 8/20 0.64
OPRK1 P41145 6/20 0.64
OPRD1 P41143 6/20 0.64
ADRB1 P08588 1/20 0.64
PDE4D Q08499 1/20 0.64
PDE3A Q14432 1/20 0.64
CTDSP1 Q9GZU7 1/20 0.63
SLC18A3 Q16572 1/20 0.58
SLC22A1 O15245 1/20 0.47
ADRA2A P08913 1/20 0.47
ARRB1 P49407 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Norcodeine SCHEMBL120271 1.00 MRGPRX2 (1.00) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL29776979 1.00 MRGPRX2 (1.00) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL18462800 1.00 MRGPRX2 (1.00) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL16922132 1.00 MRGPRX2 (1.00) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL12638889 1.00 MRGPRX2 (1.00) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL24541888 1.00 MRGPRX2 (1.00) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL4856570 0.99 MRGPRX2 (0.98) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL6220787 0.99 MRGPRX2 (0.98) MRGPRX2MAPTOPRM1OPRK1OPRD1
Norcodeine SCHEMBL7593070 0.98 MRGPRX2 (0.96) MRGPRX2MAPTOPRM1OPRK1OPRD1
Codeine SCHEMBL20703798 0.90 OPRM1 (0.83) MRGPRX2MAPTOPRM1OPRK1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1008 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118871420-A Process for the preparation of codeine, its derivatives and intermediates 暨南大学 2024-10-29 CN claimed
US-20240209403-A1 METHODS OF PRODUCING MORPHINAN ALKALOIDS AND DERIVATIVES HERCULES CAPITAL, INC., AS AGENT 2024-06-27 US claimed
US-20240165022-A1 Pharmaceutical Formulation KLARIA PHARMA HOLDING AB (SE) 2024-05-23 US claimed
US-11904049-B2 Pharmaceutical formulation KLARIA PHARMA HOLDING AB (SE) 2024-02-20 US claimed
WO-2023164889-A1 METHOD FOR PREPARING CODEINE AND DERIVATIVE AND INTERMEDIATE THEREOF 暨南大学 2023-09-07 WO claimed
CN-116660543-A Diagnostic and prognostic markers for nonalcoholic fatty liver disease and uses thereof 中国人民解放军陆军军医大学第一附属医院 2023-08-29 CN claimed
CN-116670170-A Use of LEPR agonists for pain 瑞泽恩制药公司 2023-08-29 CN claimed
EP-4214232-A2 USE OF LEPR AGONISTS FOR PAIN Regeneron Pharmaceuticals, Inc. (US) 2023-07-26 EP claimed
CN-116217641-A Synthesis method of morphine-D3-6-beta-D-glucuronide and intermediate compound thereof 上海原思标物科技有限公司 2023-06-06 CN claimed
EP-2633305-B1 AUTOMATED SYSTEM FOR SAMPLE PREPARATION AND ANALYSIS THERMO FISHER SCIENTIFIC OY (FI) 2023-03-01 EP claimed
WO-1999002529-A1 PREPARATION OF OXYMORPHONE, OXYCODONE AND DERIVATIVES PENICK CORPORATION (US) 1999-01-21 WO claimed
CN-1196955-A Thebaica giving-up vaccinum for man KUNMING BIOLOG TECH ENGINEERIN (CN) 1998-10-28 CN claimed
JP-2694156-B2 US HEALTH (US) 1997-12-24 JP claimed
EP-0496830-A4 TOTAL SYNTHESIS OF NORTHEBAINE, NORMORPHINE, NOROXYMORPHONE ENANTIOMERS AND DERIVATIVES VIA N-NOR INTERMEDIATES US HEALTH (US) 1992-09-30 EP claimed
EP-0496830-A1 TOTAL SYNTHESIS OF NORTHEBAINE, NORMORPHINE, NOROXYMORPHONE ENANTIOMERS AND DERIVATIVES VIA N-NOR INTERMEDIATES THE UNITED STATES OF AMERICA as represented by the Secretary UNITED STATES DEPARTMENT OF COMMERCE (US) 1992-08-05 EP claimed
EP-0261148-B1 ORALLY ACTIVE NONADDICTING ANALGESICS SRI INTERNATIONAL (US) 1992-01-02 EP claimed
WO-1991005768-A1 TOTAL SYNTHESIS OF NORTHEBAINE, NORMORPHINE, NOROXYMORPHONE ENANTIOMERS AND DERIVATIVES VIA N-NOR INTERMEDIATES THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, UNITED STATES DEPARTMENT OF COMMERCE (US) 1991-05-02 WO claimed
US-4940586-A Skin permeation enhancer compositions using sucrose esters ALZA CORPORATION (US) 1990-07-10 US claimed
EP-0261148-A1 ORALLY ACTIVE NONADDICTING ANALGESICS. STANFORD RES INST INT (US) 1988-03-30 EP claimed
WO-1987005903-A2 ORALLY ACTIVE NONADDICTING ANALGESICS SRI INTERNATIONAL (US) 1987-10-08 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11904049-B2 Pharmaceutical formulation OGFR, OPRL1, OPRM1 MRGPRX2 15/4885MAPT 1459/4885OPRM1 3/4885
US-20240165022-A1 Pharmaceutical Formulation OGFR, OPRL1, OPRM1 MRGPRX2 15/4885MAPT 1459/4885OPRM1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.