SCHEMBL12045337

SCHEMBL12045337

O=C(CNNCC(=O)OC(=O)C(F)(F)F)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.46
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PAM P19021 1/20 0.37
CES2 O00748 1/20 0.37
AKR1B1 P15121 1/20 0.37
PPID Q08752 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
TSHR P16473 1/20 0.36
KDM4E B2RXH2 1/20 0.35
LMNA P02545 1/20 0.35
CNR2 P34972 2/20 0.35
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9945858 0.81 CES1 (0.58) CES1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL27369755 0.72 TDP1 (0.58) CES1ALDH1A1MAPK1KMT2AHDAC8
Water SCHEMBL27403515 0.71 TDP1 (0.56) CES1ALDH1A1MAPK1KMT2AHDAC8
SCHEMBL4658964 0.70 CES1 (0.47) CES1ALDH1A1MAPK1L3MBTL1TSHR
SCHEMBL4753311 0.70 CES1 (0.71) CES1L3MBTL1CES2AKR1B1MEN1
Trifluoroacetic Acid SCHEMBL27623336 0.67 CES1 (0.56) CES1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL5150815 0.67 HDAC8 (0.57) CES1ALDH1A1MAPK1L3MBTL1CES2
SCHEMBL51367 0.66 CES1 (0.64) CES1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL27694802 0.66 ALDH1A1 (0.50) CES1ALDH1A1MAPK1L3MBTL1MEN1
SCHEMBL8052310 0.66 CES1 (0.65) CES1CRHBPCRHR2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110319594-A1 METHOD FOR PRODUCING BIVALIRUDIN SHANGHAI AMBIOPHARM, INC. (CN) 2011-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110319594-A1 METHOD FOR PRODUCING BIVALIRUDIN ARGLU1, SERPINC1, PSMA6 CES1 4402/4885CRHBP 231/4885CRHR2 1183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.