SCHEMBL1205947

SCHEMBL1205947

CCCN(CCC)Cc1ccc(NC(=O)c2ccc(CNC(=O)OC(C)(C)C)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.58
HDAC1 Q13547 4/20 0.49
HDAC6 Q9UBN7 1/20 0.48
MAPT P10636 5/20 0.48
TDP1 Q9NUW8 3/20 0.48
RORC P51449 4/20 0.47
NPSR1 Q6W5P4 2/20 0.45
XBP1 P17861 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
EPHX2 P34913 2/20 0.45
NR1H4 Q96RI1 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23899245 0.87 NAMPT (0.72) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL23899122 0.85 NAMPT (0.66) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL1637610 0.84 NAMPT (0.46) NAMPTHDAC1MAPTTDP1RORC
SCHEMBL12894119 0.83 MCHR1 (0.46) HDAC1HDAC6MAPTRORCNR1H4
SCHEMBL24891652 0.83 NAMPT (0.66) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24891860 0.82 NAMPT (0.65) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL2213535 0.82 NAMPT (0.65) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24891764 0.82 NAMPT (0.65) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL24670224 0.82 NAMPT (0.65) NAMPTHDAC1HDAC6MAPTTDP1
SCHEMBL3462770 0.80 NAMPT (0.66) NAMPTHDAC1HDAC6MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110172212-A1 AMINE-BASED COMPOUND AND USE THEREOF KUREHA CORPORATION (JP) 2011-07-14 US disclosed
US-7932281-B2 Amine-based compound and use thereof KUREHA CORPORATION (JP) 2011-04-26 US disclosed
US-20110046113-A1 AMINE COMPOUND AND USE THEREOF KUREHA CORPORATION (JP) 2011-02-24 US disclosed
US-7833991-B2 For use as antimetastatic agent or antiviral agent for HIV infection; N-(4-dipropylaminomethylphenyl)-4-{[(1H-imidazol-2-ylmethyl)-(1-methyl-1H-imidazol-2-ylmethyl)-amino]-methyl}-benzamide; chemokine receptor CXCR4 antagonists KUREHA CORPORATION (JP) 2010-11-16 US disclosed
US-20070208007-A1 Amine-Based Compound and Use Thereof KUREHA CORPORATION (JP) 2007-09-06 US disclosed
US-20070208033-A1 For use as antimetastatic agent or antiviral agent for HIV infection; N-(4-dipropylaminomethylphenyl)-4-{[(1H-imidazol-2-ylmethyl)-(1-methyl-1H-imidazol-2-ylmethyl)-amino]-methyl}-benzamide; chemokine receptor CXCR4 antagonists KUREHA CORPORATION (JP) 2007-09-06 US disclosed
US-7176227-B2 For example, N-(4-{[bis(1H-imidazol-2-ylmethyl)-amino]-methyl}-benzyl)-N',N'-dipropylbutane-1,4-diamine; efficacious against diseases such as infection with HIV virus, rheumatism, and cancer metastasis KUREHA CORPORATION (JP) 2007-02-13 US disclosed
US-20050165063-A1 Amine compounds and use thereof KUREHA CHEMICAL INDUSTRY COMPANY, LIMITED. (JP) 2005-07-28 US disclosed
EP-1550657-A1 AMINE COMPOUNDS AND USE THEREOF Kureha Chemical Industry Co., Ltd. (JP) 2005-07-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110172212-A1 AMINE-BASED COMPOUND AND USE THEREOF NR0B2, NR5A2, NR1D2 NAMPT 2707/4885HDAC1 582/4885HDAC6 1347/4885
US-20050165063-A1 Amine compounds and use thereof NR0B2, NR5A2, NR1H4 NAMPT 1941/4885HDAC1 223/4885HDAC6 1128/4885
US-20110046113-A1 AMINE COMPOUND AND USE THEREOF NR0B2, NR1D2, NR0B1 NAMPT 2324/4885HDAC1 269/4885HDAC6 1577/4885
US-20070208007-A1 Amine-Based Compound and Use Thereof NR0B2, NR5A2, NR2E1 NAMPT 2306/4885HDAC1 366/4885HDAC6 1263/4885
US-20070208033-A1 For use as antimetastatic agent or antiviral agent for HIV infection; N-(4-dipropylaminomethylphenyl)-4-{[(1H-imidazol-2-ylmethyl)-(1-methyl-1H-imidazol-2-ylmethyl)-amino]-methyl}-benzamide; chemokine receptor CXCR4 antagonists CXCR4, CXCR6, CCR5 NAMPT 1499/4885HDAC1 149/4885HDAC6 647/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.