SCHEMBL12112136

SCHEMBL12112136

CC(=O)CCC(=O)Nc1ccc(S(=O)(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)cc1

nearest known ligand 0.87

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S100B P04271 1/20 0.87
ALDH1A1 P00352 5/20 0.64
KMT2A Q03164 3/20 0.62
MEN1 O00255 2/20 0.62
TP53 P04637 1/20 0.57
GAA P10253 1/20 0.57
POLB P06746 1/20 0.56
F2 P00734 1/20 0.56
TSHR P16473 1/20 0.56
MAPT P10636 1/20 0.55
HSD17B10 Q99714 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1304849 0.93 S100B (1.00) S100BALDH1A1KMT2AMEN1TP53
SCHEMBL12112149 0.83 S100B (0.72) S100BALDH1A1KMT2AMEN1TP53
SCHEMBL12112151 0.77 ALDH1A1 (0.81) S100BALDH1A1KMT2AMEN1TP53
SCHEMBL6466850 0.72 GAA (1.00) ALDH1A1KMT2AMEN1GAAPOLB
SCHEMBL19334500 0.72 ALDH1A1 (0.67) ALDH1A1KMT2AMEN1TP53TSHR
SCHEMBL5050992 0.71 TSHR (0.76) ALDH1A1KMT2AMEN1TP53GAA
SCHEMBL11887626 0.71 TSHR (0.71) ALDH1A1GAAPOLBF2TSHR
SCHEMBL28880300 0.71 TSHR (0.81) ALDH1A1KMT2AMEN1TP53GAA
SCHEMBL14428441 0.71 FPR2 (0.88) ALDH1A1KMT2AMEN1POLBTSHR
SCHEMBL28880361 0.70 KDM4E (1.00) ALDH1A1KMT2AMEN1TP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8053477-B2 Including but hot limited to pentamidine and derivatives thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2011-11-08 US disclosed