SCHEMBL12112151

SCHEMBL12112151

Cc1c(NS(=O)(=O)c2ccc(N)cc2)c(=O)n(-c2ccccc2)n1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.81
KMT2A Q03164 3/20 0.77
MEN1 O00255 2/20 0.77
TSHR P16473 1/20 0.66
S100B P04271 1/20 0.63
TP53 P04637 1/20 0.63
LMNA P02545 3/20 0.62
GAA P10253 2/20 0.60
KDM4E B2RXH2 2/20 0.60
MAPT P10636 1/20 0.60
CASP1 P29466 1/20 0.60
HTT P42858 1/20 0.60
CASP7 P55210 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19334500 0.79 ALDH1A1 (0.67) ALDH1A1KMT2AMEN1TSHRTP53
SCHEMBL1304849 0.78 S100B (1.00) ALDH1A1KMT2AMEN1TSHRS100B
SCHEMBL12112149 0.78 S100B (0.72) ALDH1A1KMT2AMEN1TSHRS100B
SCHEMBL12112136 0.77 S100B (0.87) ALDH1A1KMT2AMEN1TSHRS100B
SCHEMBL31454744 0.76 MAPT (0.83) ALDH1A1KMT2AMEN1TSHRTP53
SCHEMBL1788374 0.76 ALDH1A1 (1.00) ALDH1A1KMT2AMEN1TSHRTP53
SCHEMBL17702679 0.76 PKM (0.68) ALDH1A1KMT2AMEN1TSHRTP53
Aminopyrine SCHEMBL7042293 0.75 ALOX15 (0.71) ALDH1A1KMT2AMEN1TSHRLMNA
SCHEMBL6466850 0.75 GAA (1.00) ALDH1A1KMT2AMEN1TSHRLMNA
SCHEMBL16134725 0.75 PKM (0.67) ALDH1A1KMT2AMEN1TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8053477-B2 Including but hot limited to pentamidine and derivatives thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2011-11-08 US disclosed
US-8053477-B2 Including but hot limited to pentamidine and derivatives thereof UNIVERSITY OF MARYLAND, BALTIMORE (US) 2011-11-08 US disclosed