SCHEMBL12200085

SCHEMBL12200085

CCC1(N)C=C(c2ccccc2)C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 8/20 0.39
MAOA P21397 8/20 0.39
MAOB P27338 8/20 0.39
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21242653 0.77 NPC1 (0.43) KDM1AMAOAMAOBNPC1RAB9A
Methane SCHEMBL28832437 0.74 NPC1 (0.36) KDM1AMAOAMAOBNPC1RAB9A
Methane SCHEMBL28950908 0.71 KDM1A (0.30) KDM1AMAOAMAOB
Methane SCHEMBL28793204 0.68 NPC1 (0.40) KDM1AMAOAMAOBNPC1RAB9A
SCHEMBL6863747 0.67 MAOA (0.37) KDM1AMAOAMAOBNPC1RAB9A
SCHEMBL14491867 0.64 NPC1 (0.43) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL28096454 0.64 NPC1 (0.47) NPC1RAB9AALDH1A1LMNAHPGD
SCHEMBL21523846 0.63 SIGMAR1 (0.41) NPC1RAB9AALDH1A1LMNAHPGD
Biphenyl SCHEMBL4840882 0.62 ALDH1A1 (0.60) MAOAALDH1A1HPGDSLC6A4
Biphenyl SCHEMBL27882978 0.62 ALDH1A1 (0.60) MAOAALDH1A1HPGDSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8329676-B2 Cycloalkane-containing sphingosine 1-phosphate agonists UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2012-12-11 US disclosed
US-20110245204-A1 CYCLOALKANE-CONTAINING SPHINGOSINE 1-PHOSPHATE AGONISTS UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2011-10-06 US disclosed
US-20100112037-A1 S1P RECEPTOR AGONISTS FOR THE TREATMENT OF CEREBRAL MALARIA LEXICON PHARMACEUTICALS, INC. 2010-05-06 US disclosed
US-20090062238-A1 METHOD FOR TREATMENT OF NEUROPATHIC PAIN UNIVERSITY OF VIRGINIA PATENT FOUNDATION 2009-03-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110245204-A1 CYCLOALKANE-CONTAINING SPHINGOSINE 1-PHOSPHATE AGONISTS S1PR1, S1PR3, S1PR4 KDM1A 3861/4885MAOA 4442/4885MAOB 4321/4885
US-20100112037-A1 S1P RECEPTOR AGONISTS FOR THE TREATMENT OF CEREBRAL MALARIA S1PR1, S1PR2, S1PR3 KDM1A 3270/4885MAOA 2782/4885MAOB 2111/4885
US-20090062238-A1 METHOD FOR TREATMENT OF NEUROPATHIC PAIN S1PR2, S1PR1, S1PR4 KDM1A 3357/4885MAOA 2859/4885MAOB 2423/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.