SCHEMBL12366175

SCHEMBL12366175

[C-]#[N+]CC(=O)NCc1cc(C)ccc1C

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
P2RX7 Q99572 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.42
KDM4C Q9H3R0 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
SETDB1 Q15047 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
TP53 P04637 1/20 0.37
POLB P06746 2/20 0.37
HPGD P15428 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366130 0.88 NPC1 (0.56) NPC1RAB9AP2RX7L3MBTL1SMN1; SMN2
SCHEMBL12366090 0.81 ALDH1A1 (0.57) NPC1RAB9AP2RX7L3MBTL1SMN1; SMN2
SCHEMBL12366100 0.78 ALDH1A1 (0.56) NPC1RAB9AL3MBTL1SMN1; SMN2LMNA
SCHEMBL12366176 0.77 NR1H4 (0.46) NPC1RAB9AL3MBTL1LMNAHTT
SCHEMBL12366162 0.77 P2RX7 (0.54) NPC1RAB9AP2RX7SMN1; SMN2ALDH1A1
SCHEMBL12366093 0.76 MMP13 (0.52) NPC1RAB9ASMN1; SMN2LMNAALDH1A1
SCHEMBL12366173 0.76 P2RX7 (0.52) NPC1RAB9AP2RX7L3MBTL1KDM4C
SCHEMBL2264102 0.76 NPC1 (0.52) NPC1RAB9AP2RX7L3MBTL1KDM4C
SCHEMBL11872322 0.76 NPC1 (0.52) NPC1RAB9AP2RX7L3MBTL1KDM4C
SCHEMBL1520513 0.76 NPC1 (0.59) NPC1RAB9AP2RX7L3MBTL1KDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed