SCHEMBL12366173

SCHEMBL12366173

[C-]#[N+]CC(=O)NCc1cccc(C)c1C

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.52
TP53 P04637 1/20 0.45
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
KDM4C Q9H3R0 1/20 0.41
HTT P42858 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366090 0.88 ALDH1A1 (0.57) P2RX7TP53ALDH1A1HPGDSMN1; SMN2
SCHEMBL3921086 0.81 P2RX7 (0.57) P2RX7TP53ALDH1A1HPGDSMN1; SMN2
SCHEMBL935059 0.79 HPGD (0.54) P2RX7TP53ALDH1A1HPGDKMT2A
SCHEMBL5670334 0.77 P2RX7 (0.52) P2RX7TP53ALDH1A1HPGDKMT2A
SCHEMBL12366130 0.76 NPC1 (0.56) P2RX7ALDH1A1SMN1; SMN2KMT2APOLB
SCHEMBL12366179 0.76 P2RX7 (0.46) P2RX7ALDH1A1HPGDSMN1; SMN2KMT2A
SCHEMBL2267520 0.76 MCL1 (0.54) P2RX7TP53ALDH1A1HPGDSMN1; SMN2
SCHEMBL12366175 0.76 NPC1 (0.56) P2RX7TP53ALDH1A1HPGDSMN1; SMN2
SCHEMBL12366196 0.76 KMT2A (0.58) P2RX7HPGDSMN1; SMN2KMT2AMEN1
SCHEMBL27847330 0.76 P2RX7 (0.51) P2RX7TP53ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed