SCHEMBL12366192

SCHEMBL12366192

[C-]#[N+]CC(=O)NCc1ccc(C(C)(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 11/20 0.54
NR1H4 Q96RI1 9/20 0.54
HDAC3 O15379 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
RAB9A P51151 2/20 0.51
LMNA P02545 1/20 0.51
ALDH1A1 P00352 1/20 0.51
NPC1 O15118 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366117 0.84 HDAC1 (0.56) EPHX2HDAC3HDAC8HDAC6RAB9A
SCHEMBL19513354 0.82 EPHX2 (0.62) EPHX2NR1H4HDAC3HDAC8HDAC6
SCHEMBL12366188 0.82 LMNA (0.47) KMT2ALMNAALDH1A1
SCHEMBL12366100 0.82 ALDH1A1 (0.56) MEN1KMT2ARAB9ALMNAALDH1A1
SCHEMBL12993441 0.80 EPHX2 (0.59) EPHX2NR1H4HDAC3HDAC8HDAC6
SCHEMBL5178356 0.80 EPHX2 (0.64) EPHX2NR1H4HDAC3HDAC8HDAC6
SCHEMBL3421393 0.79 MEN1 (0.60) EPHX2NR1H4HDAC3HDAC8HDAC6
SCHEMBL12366096 0.79 L3MBTL1 (0.57) MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL12366142 0.79 KMT2A (0.59) MEN1KMT2ACYP2C19RAB9AALDH1A1
SCHEMBL249685 0.79 EPHX2 (0.62) EPHX2NR1H4HDAC3HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed