SCHEMBL12366117

SCHEMBL12366117

[C-]#[N+]CC(=O)NCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.56
HDAC8 Q9BY41 2/20 0.56
HDAC3 O15379 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC10 Q969S8 1/20 0.56
HDAC11 Q96DB2 1/20 0.56
HDAC6 Q9UBN7 1/20 0.56
MTOR P42345 2/20 0.50
P2RX7 Q99572 2/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
LSS P48449 1/20 0.49
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MAPK14 Q16539 1/20 0.47
NAMPT P43490 1/20 0.47
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12366192 0.84 EPHX2 (0.54) HDAC8HDAC3HDAC6NPC1RAB9A
SCHEMBL12366113 0.82 L3MBTL1 (0.63) NPC1RAB9AMAPK14LMNAPOLB
SCHEMBL12366135 0.82 LMNA (0.62) CA12CA1CA2NPC1RAB9A
SCHEMBL12366146 0.81 EPHX2 (0.53) CA12CA1CA2CA7NAMPT
SCHEMBL12366188 0.79 LMNA (0.47) CA12CA1CA2CA7LMNA
SCHEMBL12366096 0.79 L3MBTL1 (0.57) CA12CA1CA2CA7POLB
SCHEMBL10594986 0.79 HDAC3 (0.60) HDAC1HDAC8HDAC3HDAC2HDAC10
SCHEMBL6366481 0.79 ALDH1A1 (0.57) RAB9ALMNAALDH1A1
SCHEMBL934145 0.79 HDAC3 (0.60) HDAC1HDAC8HDAC3HDAC2HDAC10
SCHEMBL12366142 0.79 KMT2A (0.59) CA12CA1CA2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed