SCHEMBL12368809

SCHEMBL12368809

CN1CCN(c2ccccc2CO)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 2/20 0.61
DRD2 P14416 3/20 0.58
DRD3 P35462 3/20 0.58
HTR1A P08908 1/20 0.58
DRD4 P21917 1/20 0.58
HTR2A P28223 1/20 0.58
HTR2C P28335 1/20 0.58
ADRA2C P18825 1/20 0.55
EGFR P00533 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45
BRD4 O60885 2/20 0.45
BRPF1 P55201 2/20 0.45
BRD9 Q9H8M2 2/20 0.45
HTR6 P50406 1/20 0.45
BRD7 Q9NPI1 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10711290 0.98 NCF1 (0.59) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL4960474 0.90 KDM4E (0.52) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL5722525 0.86 NCF1 (0.58) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL8361520 0.85 DRD2 (0.72) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL18756992 0.83 HTR1A (0.53) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL721985 0.82 NCF1 (0.49) NCF1MAPK1KMT2AKDM4EALDH1A1
SCHEMBL29505669 0.81 NCF1 (0.87) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL110927 0.81 NCF1 (0.87) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL14355759 0.81 NCF1 (0.61) NCF1DRD2DRD3HTR1ADRD4
SCHEMBL5161795 0.81 NCF1 (0.61) NCF1DRD2DRD3HTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11345711-B2 8,9-dihydroimidazo[1,2-a]pyrimido[5,4-e]pyrimidin-5(6H)-ones Impact Therapeutics (Shanghai), Inc (CN) 2022-05-31 US disclosed
US-20200385394-A1 8,9-DIHYDROIMIDAZO[1,2-a]PYRIMIDO[5,4-e]PYRIMIDIN-5(6H)-ONES Impact Therapeutics (Shanghai), Inc (CN) 2020-12-10 US disclosed
US-10703759-B2 8,9-dihydroimidazo[1,2-a]pyrimido[5,4-e]pyrimidin-5(6H)-ones IMPACT THERAPEUTICS, INC (CN) 2020-07-07 US disclosed
US-20190308984-A1 8,9-DIHYDROIMIDAZO[1,2-a]PYRIMIDO[5,4-e]PYRIMIDIN-5(6H)-ONES Impact Therapeutics (Shanghai), Inc (CN) 2019-10-10 US disclosed
US-9442399-B2 Electrophotographic photosensitive member, process cartridge, electrophotographic apparatus and phthalocyanine crystal CANON KABUSHIKI KAISHA (JP) 2016-09-13 US disclosed
US-9442399-B2 Electrophotographic photosensitive member, process cartridge, electrophotographic apparatus and phthalocyanine crystal CANON KABUSHIKI KAISHA (JP) 2016-09-13 US disclosed
EP-2743772-B1 Electrophotographic photosensitive member, process cartridge, electrophotographic apparatus and phthalocyanine crystal CANON KK (JP) 2016-04-20 EP disclosed
US-20140170542-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS AND PHTHALOCYANINE CRYSTAL CANON KABUSHIKI KAISHA (JP) 2014-06-19 US disclosed
US-20140170542-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, ELECTROPHOTOGRAPHIC APPARATUS AND PHTHALOCYANINE CRYSTAL CANON KABUSHIKI KAISHA (JP) 2014-06-19 US disclosed
EP-2743772-A1 Electrophotographic photosensitive member, process cartridge, electrophotographic apparatus and phthalocyanine crystal Canon Kabushiki Kaisha (JP) 2014-06-18 EP disclosed
US-8530465-B2 1, 2-disubstituted amido-anthraquinone derivatives, preparation method and application thereof NATIONAL DEFENSE MEDICAL CENTER (TW) 2013-09-10 US disclosed
US-20130059862-A1 Novel 1, 2-Disubstituted Amido-anthraquinone Derivatives, Preparation Method and application thereof HUANG HSU-SHAN (TW) 2013-03-07 US disclosed
US-8304415-B2 1, 2-disubstituted amido-anthraquinone derivatives, preparation method and application thereof NATIONAL DEFENSE MEDICAL CENTER (TW) 2012-11-06 US disclosed
US-20110207739-A1 Novel 1, 2-Disubstituted Amido-anthraquinone Derivatives, Preparation Method and application thereof NATIONAL DEFENSE MEDICAL CENTER (TW) 2011-08-25 US disclosed
US-7291619-B2 Melanocortin receptor agonists ELI LILLY AND COMPANY (US) 2007-11-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190308984-A1 8,9-DIHYDROIMIDAZO[1,2-a]PYRIMIDO[5,4-e]PYRIMIDIN-5(6H)-ONES WEE1, WEE2, CCNE1 NCF1 3087/4885DRD2 4463/4885DRD3 4251/4885
US-11345711-B2 8,9-dihydroimidazo[1,2-a]pyrimido[5,4-e]pyrimidin-5(6H)-ones WEE1, WEE2, CCNE1 NCF1 3087/4885DRD2 4463/4885DRD3 4251/4885
US-10703759-B2 8,9-dihydroimidazo[1,2-a]pyrimido[5,4-e]pyrimidin-5(6H)-ones WEE1, WEE2, CCNE1 NCF1 3087/4885DRD2 4463/4885DRD3 4251/4885
US-20110207739-A1 Novel 1, 2-Disubstituted Amido-anthraquinone Derivatives, Preparation Method and application thereof ANXA1, ANXA5, ANXA2 NCF1 1357/4885DRD2 4174/4885DRD3 3905/4885
US-20130059862-A1 Novel 1, 2-Disubstituted Amido-anthraquinone Derivatives, Preparation Method and application thereof ANXA5, ANXA1, HCCS NCF1 1351/4885DRD2 4132/4885DRD3 3867/4885
US-20200385394-A1 8,9-DIHYDROIMIDAZO[1,2-a]PYRIMIDO[5,4-e]PYRIMIDIN-5(6H)-ONES WEE1, WEE2, CCNE1 NCF1 3087/4885DRD2 4463/4885DRD3 4251/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.