SCHEMBL12377475

SCHEMBL12377475

NCC(=O)Nc1cccc(B(O)O)c1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.60
CA2 P00918 3/20 0.60
NLRP3 Q96P20 1/20 0.58
TERT O14746 1/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
TRPV1 Q8NER1 1/20 0.48
ESRRG P62508 4/20 0.45
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
ENPP2 Q13822 1/20 0.43
POLB P06746 1/20 0.42
NR4A1 P22736 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16387340 0.84 NLRP3 (0.53) CA1CA2NLRP3TERTMEN1
SCHEMBL6353539 0.83 RAB9A (0.63) NLRP3MEN1KMT2AALDH1A1POLB
SCHEMBL8622297 0.83 NLRP3 (0.58) NLRP3MEN1KMT2ATRPV1ESRRG
SCHEMBL7744399 0.83 NLRP3 (0.58) CA1CA2NLRP3MEN1KMT2A
SCHEMBL14756770 0.83 NLRP3 (0.58) CA1CA2NLRP3MEN1KMT2A
SCHEMBL7865481 0.83 L3MBTL1 (0.61) CA1CA2NLRP3MEN1KMT2A
SCHEMBL16387330 0.82 HDAC1 (0.55) NLRP3MEN1KMT2AKDM4E
Hydrochloric Acid SCHEMBL19747848 0.82 CA1 (0.67) CA1CA2TERTMEN1KMT2A
SCHEMBL1303751 0.81 TRPV1 (0.51) CA1CA2NLRP3TRPV1ESRRG
SCHEMBL1810118 0.81 L3MBTL1 (0.57) NLRP3MEN1KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7989625-B2 Thienopyridines MERCK PATENT GMBH (DE) 2011-08-02 US disclosed
US-7989625-B2 Thienopyridines MERCK PATENT GMBH (DE) 2011-08-02 US disclosed
US-20100048558-A1 THIENOPYRIDINES MERCK PATENT GESELLSCHAFT (DE) 2010-02-25 US disclosed
US-20100048558-A1 THIENOPYRIDINES MERCK PATENT GESELLSCHAFT (DE) 2010-02-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048558-A1 THIENOPYRIDINES HSP90AB2P, HSP90AB1, HSP90AA1 CA1 4694/4885CA2 2279/4885NLRP3 1125/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.