SCHEMBL12379331

SCHEMBL12379331

c1cnc2c(c1)CC1C2CCC2C3CCCCC3CCC12

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.33
HTR2A P28223 6/20 0.31
HTR2C P28335 6/20 0.31
HTR2B P41595 6/20 0.31
HRH3 Q9Y5N1 5/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29587352 0.77 HTR2A (0.36) HTR2AHTR2CHTR2BHRH3
SCHEMBL1698200 0.70 KDM4E (0.39) HTR2AHTR2CHTR2BHRH3
SCHEMBL1698216 0.69 HDAC1 (0.40)
SCHEMBL1760687 0.63 ALDH1A1 (0.47)
SCHEMBL12475384 0.63 ALDH1A1 (0.47)
SCHEMBL30631702 0.62
SCHEMBL3835964 0.62 OPRL1 (0.36)
SCHEMBL375061 0.61 ALDH1A1 (0.44)
SCHEMBL15454179 0.61 ALDH1A1 (0.44)
SCHEMBL29886257 0.61 ALDH1A1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8003783-B2 Steroid 17 beta -hydroxysteroid dehydrogenase inhibitors substituted with one or more oxime groups, especially aromatase inhibitors used in the treatment of endocrine-dependent tumors, especially breast cancer STERIX LIMITED (GB) 2011-08-23 US disclosed