SCHEMBL12420394

SCHEMBL12420394

CCc1ccc(-c2cn(-c3ccc(F)cc3)nn2)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.63
PTGS1 P23219 3/20 0.63
CA1 P00915 4/20 0.59
CA2 P00918 4/20 0.59
CA5A P35218 3/20 0.59
CA5B Q9Y2D0 3/20 0.59
S1PR1 P21453 4/20 0.57
FLT3 P36888 3/20 0.56
CA12 O43570 3/20 0.50
CA9 Q16790 3/20 0.50
S1PR3 Q99500 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16220811 0.87 PTGS2 (0.72) PTGS2PTGS1CA1CA2CA5A
SCHEMBL18031098 0.85 S1PR1 (0.60) PTGS2PTGS1CA1CA2CA5A
SCHEMBL12420291 0.85 S1PR1 (0.59) PTGS2PTGS1CA1CA2CA5A
SCHEMBL19186826 0.84 FLT3 (0.70) PTGS2PTGS1CA1CA2CA5A
SCHEMBL12420391 0.83 STS (0.59) PTGS2PTGS1CA1CA2CA5A
SCHEMBL23557718 0.80 PTGS2 (0.63) PTGS2PTGS1CA1CA2CA5A
SCHEMBL18031100 0.80 PTGS2 (0.63) PTGS2PTGS1CA1CA2CA5A
SCHEMBL28068164 0.80 PTGS2 (0.62) PTGS2PTGS1CA1CA2CA5A
SCHEMBL28337478 0.80 FLT3 (0.65) PTGS2PTGS1CA1CA2CA5A
SCHEMBL12420293 0.78 HSD17B1 (0.56) CA1CA2S1PR1FLT3CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130096165-A1 COMPOUNDS AND METHODS FOR MODULATING G PROTEIN-COUPLED RECEPTORS IRM LLC (BM) 2013-04-18 US disclosed
US-8362050-B2 Compounds and methods for modulating G protein-coupled receptors IRM LLC (BM) 2013-01-29 US disclosed
US-20110172278-A1 COMPOUNDS AND METHODS FOR MODULATING G PROTEIN-COUPLED RECEPTORS IRM LLC (BM) 2011-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130096165-A1 COMPOUNDS AND METHODS FOR MODULATING G PROTEIN-COUPLED RECEPTORS GRK2, GRK3, GPR3 PTGS2 481/4885PTGS1 440/4885CA1 4087/4885
US-20110172278-A1 COMPOUNDS AND METHODS FOR MODULATING G PROTEIN-COUPLED RECEPTORS GRK2, GRK3, GPR3 PTGS2 481/4885PTGS1 440/4885CA1 4087/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.