SCHEMBL12425650

SCHEMBL12425650

CC(C)OC(=O)N1C2CCC1CN(C(=O)c1ccc(N)nn1)C2

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPC6 Q9Y210 17/20 0.39
GPR119 Q8TDV5 2/20 0.35
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2300760 0.84 HSD11B1 (0.45) TRPC6GPR119
SCHEMBL25317444 0.73 GABRA1 (0.44) TRPC6
SCHEMBL12425603 0.71 CHRNA4 (0.40) TRPC6
SCHEMBL20929521 0.66 NPC1 (0.49) ALDH1A1
SCHEMBL12425623 0.65 CDK4 (0.49) ALDH1A1
SCHEMBL1713578 0.65 GPR119 (0.38) GPR119
SCHEMBL2298739 0.64 SPR (0.46) GPR119
SCHEMBL2300794 0.64 HDAC1 (0.52) GPR119
SCHEMBL12425428 0.64 HDAC1 (0.55) GPR119
SCHEMBL13738462 0.63 MAPK1 (0.41) GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101409-A1 PYRROLOPYRIMIDINE COMPOUNDS AS INHIBITORS OF CDK4/6 NOVARTIS AG (CH) 2011-08-25 WO disclosed