SCHEMBL12436971

SCHEMBL12436971

[C-]#[N+]CC(=O)N1CCC(C(C)=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
NPC1 O15118 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.35
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
YAP1 P46937 1/20 0.34
TEAD4 Q15561 1/20 0.34
PKM P14618 1/20 0.33
POLB P06746 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4870186 0.79 ALDH1A1 (0.37) ALDH1A1NPC1L3MBTL1SMN1; SMN2MEN1
SCHEMBL12436953 0.77 EPHX2 (0.50) ALDH1A1NPC1GAA
SCHEMBL12436034 0.77 ALDH1A1 (0.42) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL15369211 0.76 ALDH1A1 (0.41) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL14902198 0.76 ALDH1A1 (0.41) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL17812266 0.76 CPN1 (0.47) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL13804082 0.76 ALDH1A1 (0.41) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL295163 0.74 ALDH1A1 (0.50) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL13629807 0.74 ALDH1A1 (0.40) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2
SCHEMBL12436973 0.74 NAMPT (0.53) ALDH1A1NPC1L3MBTL1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME NTSR2, BDKRB1, AVPR1B ALDH1A1 3648/4885NPC1 1587/4885L3MBTL1 1003/4885
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof NTSR2, NTSR1, HNMT ALDH1A1 2667/4885NPC1 1263/4885L3MBTL1 2718/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.