SCHEMBL12445874

SCHEMBL12445874

CNC(=O)CCc1cc(NC(=O)c2cnc(-c3nccs3)cn2)ccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
BLM P54132 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MCL1 Q07820 1/20 0.36
ADORA2A P29274 5/20 0.36
SCD O00767 1/20 0.35
SCD5 Q86SK9 1/20 0.35
PRKCI P41743 1/20 0.35
TYK2 P29597 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446185 0.84 NPC1 (0.43) ALDH1A1NPC1RAB9AL3MBTL1KDM4E
SCHEMBL7941942 0.77 SORT1 (0.41) NPC1RAB9APRKCITSHRBACE1
SCHEMBL12445675 0.77 BACE1 (0.49) BACE1GRM4
SCHEMBL12446237 0.77 BACE1 (0.47) NPC1RAB9AKDM4EPRKCIHPGD
SCHEMBL12445674 0.76 BACE1 (0.47) PRKCIBACE1GRM4
SCHEMBL7933492 0.75 BACE1 (0.51) MCL1SCDSCD5PRKCIBACE1
SCHEMBL12445871 0.74 BACE1 (0.47) BACE1GRM4
SCHEMBL12445846 0.74 GRM4 (0.38) NPC1RAB9APRKCISMN1; SMN2BACE1
SCHEMBL12446239 0.72 PRKCI (0.40) ALDH1A1PRKCITYK2TSHRBACE1
SCHEMBL7943969 0.70 PRKCI (0.47) PRKCITYK2BACE1GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2360155-A1 2-AMINOPYRIDIN-4-ONE AND 2-AMINOPYRIDINE DERIVATIVE BOTH HAVING BACE1-INHIBITING ACTIVITY Shionogi & Co., Ltd. (JP) 2011-08-24 EP disclosed