SCHEMBL12445916

SCHEMBL12445916

N[C@]1(c2ccc(Cl)cc2)CN[C@@H](C(=O)NCCC2CC2)[C@@H]1c1cccc(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 9/20 0.44
TP53 P04637 3/20 0.44
MDM4 O15151 1/20 0.42
CHRM1 P11229 1/20 0.38
HSD11B1 P28845 1/20 0.36
CHRM4 P08173 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
TAAR1 Q96RJ0 2/20 0.35
GLA P06280 1/20 0.35
CNR1 P21554 1/20 0.35
CACNA1B Q00975 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446085 0.88 MDM2 (0.55) MDM2TP53MDM4HSD11B1TAAR1
SCHEMBL7948520 0.84 MDM2 (0.41) MDM2TP53MDM4HSD11B1CACNA1B
SCHEMBL12446087 0.83 MDM2 (0.44) MDM2TP53MDM4
SCHEMBL12446511 0.82 MDM2 (0.54) MDM2TP53MDM4CNR1
SCHEMBL7952593 0.81 P2RX7 (0.40) MDM2TP53MDM4
SCHEMBL12446587 0.81 LMNA (0.46) MDM2TP53CNR1
SCHEMBL18773089 0.79 MDM2 (0.60) MDM2TP53MDM4
SCHEMBL12446512 0.77 HTT (0.46) MDM2TP53MDM4HSD11B1CACNA1B
SCHEMBL12446594 0.75 LMNA (0.53) POLB
SCHEMBL7959673 0.74 MDM2 (0.46) MDM2TP53MDM4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011098398-A1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-18 WO disclosed