SCHEMBL12446512

SCHEMBL12446512

CN(C)C(=O)[C@@H]1NC[C@](N)(c2ccc(Cl)cc2)[C@H]1c1cccc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
MDM2 Q00987 9/20 0.44
TP53 P04637 5/20 0.39
SLC9A1 P19634 2/20 0.38
HSD11B1 P28845 1/20 0.38
CACNA1B Q00975 4/20 0.37
KDM1A O60341 2/20 0.36
RCOR1 Q9UKL0 2/20 0.36
MDM4 O15151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12446085 0.78 MDM2 (0.55) HTTMDM2TP53HSD11B1CACNA1B
SCHEMBL12445916 0.77 MDM2 (0.44) MDM2TP53HSD11B1CACNA1BMDM4
SCHEMBL12446107 0.76 HSD11B1 (0.39) MDM2TP53SLC9A1HSD11B1CACNA1B
SCHEMBL7948520 0.75 MDM2 (0.41) MDM2TP53HSD11B1CACNA1BMDM4
SCHEMBL18773007 0.74 MDM2 (0.64) MDM2TP53MDM4
SCHEMBL12446087 0.74 MDM2 (0.44) MDM2TP53MDM4
SCHEMBL12446511 0.73 MDM2 (0.54) HTTMDM2TP53MDM4
SCHEMBL7952593 0.73 P2RX7 (0.40) HTTMDM2TP53MDM4
SCHEMBL12446587 0.73 LMNA (0.46) HTTMDM2TP53
SCHEMBL7959673 0.72 MDM2 (0.46) MDM2TP53MDM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011098398-A1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES F. HOFFMANN-LA ROCHE AG (CH) 2011-08-18 WO disclosed