SCHEMBL1246307

SCHEMBL1246307

CCOC(=O)N(c1ccccc1Cl)c1c(-c2ccc(-c3cccc(CC(=O)O)c3)cc2)noc1C

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.44
PPARD Q03181 5/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PTGS2 P35354 1/20 0.39
GPBAR1 Q8TDU6 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SCN9A Q15858 1/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1246467 0.94 NR1H4 (0.43) NR1H4PPARDPTGS2GPBAR1SCN9A
SCHEMBL1245358 0.92 NR1H4 (0.42) NR1H4PPARDPTGS2GPBAR1SCN9A
SCHEMBL1246346 0.92 SCN9A (0.38) NR1H4PPARDGPBAR1SCN9AMAPT
SCHEMBL1245136 0.90 NR1H4 (0.38) NR1H4PPARDTDP1MAPT
SCHEMBL1246951 0.90 CYP11B1 (0.40) NR1H4PTGS2GPBAR1TDP1SCN9A
SCHEMBL1246476 0.90 NR1H4 (0.42) NR1H4PPARDGPBAR1MAPT
SCHEMBL1245176 0.89 NR1H4 (0.40) NR1H4PPARDGPBAR1SCN9AMAPT
SCHEMBL1247166 0.88 TSHR (0.44) NR1H4PPARDTSHR
SCHEMBL1247326 0.88 PPARD (0.37) NR1H4PPARDGPBAR1SCN9AMAPT
SCHEMBL1245320 0.88 NR1H4 (0.45) NR1H4PTGS2GPBAR1TDP1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed