SCHEMBL1246951

SCHEMBL1246951

CCOC(=O)N(c1ccccc1Cl)c1c(-c2ccc(-c3cncc(CC(=O)O)c3)cc2)noc1C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
LPAR1 Q92633 1/20 0.37
LPAR2 Q9HBW0 1/20 0.37
LPAR3 Q9UBY5 1/20 0.37
GPBAR1 Q8TDU6 4/20 0.36
NR1H4 Q96RI1 3/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
HPGD P15428 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP2C19 P33261 1/20 0.35
SCN9A Q15858 2/20 0.35
PTGS2 P35354 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1245358 0.90 NR1H4 (0.42) LPAR1LPAR2LPAR3GPBAR1NR1H4
SCHEMBL1246307 0.90 NR1H4 (0.44) GPBAR1NR1H4MAPTTDP1SCN9A
SCHEMBL1246467 0.87 NR1H4 (0.43) LPAR1LPAR2LPAR3GPBAR1NR1H4
SCHEMBL1245176 0.87 NR1H4 (0.40) LPAR1LPAR2LPAR3GPBAR1NR1H4
SCHEMBL3707597 0.87 LPAR1 (0.46) CYP11B1CYP11B2LPAR1LPAR2LPAR3
SCHEMBL1246476 0.86 NR1H4 (0.42) LPAR1LPAR2LPAR3GPBAR1NR1H4
SCHEMBL1246477 0.85 NR1H4 (0.42) GPBAR1NR1H4MAPTALDH1A1
SCHEMBL1246346 0.85 SCN9A (0.38) GPBAR1NR1H4MAPTALDH1A1SCN9A
SCHEMBL1247748 0.85 SCN9A (0.39) GPBAR1NR1H4MAPTALDH1A1POLB
SCHEMBL1245136 0.84 NR1H4 (0.38) NR1H4MAPTALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed