SCHEMBL12466708

SCHEMBL12466708

O=CN(OCC1c2ccccc2-c2ccccc21)C(CCCCCC(=O)O)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.49
CASP3 P42574 3/20 0.37
TBXA2R P21731 1/20 0.35
CYP1A2 P05177 1/20 0.34
TSHR P16473 1/20 0.34
FABP7 O15540 2/20 0.34
FABP5 Q01469 2/20 0.34
TLR2 O60603 2/20 0.33
TBXAS1 P24557 1/20 0.33
EGFR P00533 1/20 0.33
ACLY P53396 2/20 0.33
FOLH1 Q04609 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4740141 0.88 KMT2A (0.38) KMT2ACASP3CYP1A2TSHRFABP7
SCHEMBL27527132 0.87 CASP3 (0.38) KMT2ACASP3FABP7FABP5TLR2
SCHEMBL29277349 0.78 KMT2A (0.55) KMT2ACASP3FABP7FABP5TLR2
SCHEMBL29277350 0.78 KMT2A (0.55) KMT2ACASP3FABP7FABP5TLR2
SCHEMBL27042592 0.77 CASP3 (0.35) KMT2ACASP3CYP1A2TSHRFABP7
SCHEMBL289035 0.77 FABP5 (0.40) KMT2ACASP3CYP1A2TSHRFABP7
SCHEMBL1557276 0.74 PPARG (0.41) KMT2ACASP3
SCHEMBL1556697 0.74 OPRM1 (0.38) KMT2ACASP3
SCHEMBL5972005 0.73 KMT2A (0.70) KMT2ACASP3FABP7FABP5EGFR
SCHEMBL2401694 0.73 KMT2A (0.70) KMT2ACASP3FABP7FABP5EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103328-A1 LABELED, NON- PEPTIDIC MULTIVALENT INTEGRIN ALPHA -V - BETA - 3 ANTAGONISTS, COMPOSITIONS CONTAINING THEM AND THEIR USE THE METHODIST HOSPITAL RESEARCH INSTITUTE (US) 2012-08-02 WO disclosed