SCHEMBL12466749

SCHEMBL12466749

COc1cccc(-c2conc2C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
PIN1 Q13526 1/20 0.52
GPR35 Q9HC97 3/20 0.46
EGLN1 Q9GZT9 1/20 0.46
IKBKB O14920 1/20 0.45
NPC1 O15118 1/20 0.45
TP53 P04637 1/20 0.45
NFKB1 P19838 1/20 0.45
RAB9A P51151 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
TDO2 P48775 1/20 0.45
PRKAB2 O43741 1/20 0.44
PRKAG1 P54619 1/20 0.44
PRKAA2 P54646 1/20 0.44
PRKAA1 Q13131 1/20 0.44
PRKAG3 Q9UGI9 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28827222 0.82 ALDH1A1 (0.50) ALDH1A1HPGDEGLN1SMN1; SMN2PRKAB2
SCHEMBL4075531 0.78 PTPN1 (0.47) ALDH1A1PIN1SMN1; SMN2PTPN1LMNA
SCHEMBL28069539 0.78 MCL1 (0.44) ALDH1A1HPGDPTPN1LMNA
SCHEMBL28192178 0.76 PIN1 (0.56) ALDH1A1HPGDPIN1GPR35SMN1; SMN2
SCHEMBL1870966 0.76 DYRK1A (0.54) ALDH1A1HPGDPIN1TDP1PRKAB2
SCHEMBL8202718 0.75 PRKAB2 (0.55) ALDH1A1HPGDGPR35SMN1; SMN2PRKAB2
SCHEMBL16134763 0.75 POLB (0.52) ALDH1A1NPC1RAB9ASMN1; SMN2LMNA
SCHEMBL19207037 0.74 LMNA (0.51) ALDH1A1HPGDPIN1EGLN1NPC1
SCHEMBL1167103 0.72 GSK3B (0.61) ALDH1A1HPGDPIN1IKBKBNR1H2
SCHEMBL22619671 0.72 MKNK1 (0.50) ALDH1A1GPR35IKBKBTP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103113-A1 PYRAZINE AND IMIDAZOLIDINE DERIVATIVES AND THEIR USES TO TREAT HEPATITIS C GILEAD PHARMASSET, LLC (US) 2012-08-02 WO disclosed