SCHEMBL28192178

SCHEMBL28192178

COc1cccc(-c2c[nH]nc2C(=O)O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.56
LMNA P02545 3/20 0.51
ALDH1A1 P00352 2/20 0.51
PRKAB2 O43741 1/20 0.51
PRKAG1 P54619 1/20 0.51
PRKAA2 P54646 1/20 0.51
PRKAA1 Q13131 1/20 0.51
PRKAG3 Q9UGI9 1/20 0.51
PRKAG2 Q9UGJ0 1/20 0.51
PRKAB1 Q9Y478 1/20 0.51
HPGD P15428 1/20 0.50
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PLK1 P53350 1/20 0.47
GRK6 P43250 1/20 0.45
NR1H2 P55055 2/20 0.45
NR1H3 Q13133 2/20 0.45
AKR1C3 P42330 1/20 0.45
AKR1C2 P52895 1/20 0.45
NOTUM Q6P988 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28191526 0.87 MAPT (0.56) PIN1LMNAALDH1A1PRKAB2PRKAG1
SCHEMBL9353501 0.82 PRKAG1 (0.53) ALDH1A1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL948199 0.80 KDM4E (0.50) PIN1LMNAALDH1A1PRKAB2PRKAG1
SCHEMBL10432377 0.79 PIN1 (0.52) PIN1PLK1GRK6NOTUMGPR35
SCHEMBL4700185 0.77 TDO2 (0.55) LMNAALDH1A1NR1H2NR1H3NOTUM
SCHEMBL1870966 0.77 DYRK1A (0.54) PIN1LMNAALDH1A1PRKAB2PRKAG1
SCHEMBL12466749 0.76 ALDH1A1 (0.56) PIN1LMNAALDH1A1PRKAB2PRKAG1
SCHEMBL15995331 0.76 ROCK1 (0.68) DYRK1A
SCHEMBL16109091 0.76 KDM4E (0.36) PIN1LMNAALDH1A1PRKAB2PRKAG1
SCHEMBL15510700 0.76 KDM4E (0.40) PIN1LMNAALDH1A1PRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107406427-A Alkynyl alcohols and methods of use thereof 豪夫迈·罗氏有限公司 2017-11-28 CN disclosed