SCHEMBL1246796

SCHEMBL1246796

CCN(C(=O)O)c1cccc2c1OCCN2

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.36
HTR1A P08908 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
AKT1 P31749 1/20 0.34
ALDH1A1 P00352 3/20 0.34
TSHR P16473 2/20 0.34
GLA P06280 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
MAPK14 Q16539 1/20 0.32
MAPT P10636 2/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31
AR P10275 1/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971530 0.79 TP53 (0.50) ALDH1A1TSHRGLAKDM4EMAPK14
SCHEMBL9911042 0.76 ADORA2A (0.43) DRD2HTR1AADORA2AADORA1AKT1
Propionic Acid SCHEMBL2687317 0.75 DRD2 (0.40) DRD2HTR1AADORA2AADORA1AKT1
Propionic Acid SCHEMBL2686240 0.74 NOTUM (0.41) DRD2HTR1AADORA2AADORA1AKT1
Propionic Acid SCHEMBL2637824 0.74 ADORA2A (0.45) DRD2HTR1AADORA2AADORA1AKT1
SCHEMBL10748058 0.73 HPGD (0.41) ALDH1A1TSHRGLAKDM4EMAPT
SCHEMBL1340046 0.72 ALOX5 (0.40) DRD2HTR1AADORA2AADORA1AKT1
SCHEMBL18665582 0.71 KDM4E (0.43) DRD2HTR1AADORA2AADORA1AKT1
SCHEMBL1612190 0.70 TSHR (0.49) ALDH1A1TSHRMAPTGAAHSD17B10
SCHEMBL1549847 0.70 ADRA1D (0.43) ADORA2AADORA1AKT1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459572-A2 SPIROCYCLIC AMIDE DERIVATIVES AstraZeneca AB (SE) 2012-06-06 EP disclosed
WO-2011012896-A2 COMPOUNDS - 801 ASTRAZENECA AB (SE) 2011-02-03 WO disclosed