SCHEMBL12468753

SCHEMBL12468753

Fc1cccc(F)c1Cn1ccnn1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.55
CA5A P35218 1/20 0.45
KEAP1 Q14145 1/20 0.39
CCR1 P32246 1/20 0.38
CCR2 P41597 1/20 0.38
ALDH1A1 P00352 2/20 0.37
DPP4 P27487 1/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29820003 0.80 CYP19A1 (0.70) CYP19A1CCR1CCR2ALDH1A1KDM4E
SCHEMBL12468869 0.80 CYP19A1 (0.70) CYP19A1CCR1CCR2ALDH1A1KDM4E
SCHEMBL12468796 0.79 CYP19A1 (0.50) CYP19A1CCR1CCR2DPP4
SCHEMBL7468845 0.75 CYP19A1 (0.56) CYP19A1CCR1CCR2DPP4
SCHEMBL29820311 0.74 CYP19A1 (0.64) CYP19A1KEAP1CCR1CCR2ALDH1A1
SCHEMBL28263864 0.72 CYP19A1 (0.68) CYP19A1CCR1CCR2
SCHEMBL29820189 0.72 CYP19A1 (0.67) CYP19A1CCR1CCR2ALDH1A1TSHR
SCHEMBL13201552 0.71 CYP19A1 (0.80) CYP19A1CCR1CCR2
SCHEMBL155247 0.71 CYP19A1 (1.00) CYP19A1CCR1CCR2POLB
Hydrochloric Acid SCHEMBL7263772 0.69 CYP19A1 (0.96) CYP19A1CCR1CCR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117105873-A Preparation method of rufeamide intermediate 宿州亿帆药业有限公司 2023-11-24 CN disclosed
CN-117050027-A Preparation method of rufeamide impurity reference substance 宿州亿帆药业有限公司 2023-11-14 CN disclosed
CN-110072521-A Pharmaceutical combination comprising a T-type calcium channel blocker 爱杜西亚药品有限公司 2019-07-30 CN disclosed
CN-107406420-A Substituted triazoles and methods related thereto 纽罗克里生物科学有限公司 2017-11-28 CN disclosed
US-8969556-B2 Purine-based triazoles CASE WESTERN RESERVE UNIVERSITY (US) 2015-03-03 US disclosed
US-20140045866-A1 PURINE-BASED TRIAZOLES CASE WESTERN RESERVE UNIVERSITY 2014-02-13 US disclosed
WO-2012051296-A2 PURINE-BASED TRIAZOLES CASE WESTERN RESERVE UNIVERSITY (US) 2012-04-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140045866-A1 PURINE-BASED TRIAZOLES PNP, TK2, NME4 CYP19A1 4083/4885CA5A 1546/4885KEAP1 3890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.