SCHEMBL12469647

SCHEMBL12469647

Nc1ccc(-c2ccc(-c3ncco3)c3c2CNC3=O)c(F)c1.Nc1ccc(F)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.38
FLT3 P36888 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
ADRA1A P35348 2/20 0.33
ADRA2A P08913 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1B P35368 1/20 0.33
GRM5 P41594 1/20 0.33
GRM2 Q14416 1/20 0.33
KIT P10721 1/20 0.32
RORC P51449 1/20 0.32
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469609 0.82 BTK (0.39) BTKFLT3PDE3BPDE3AGRM2
SCHEMBL12469667 0.81 BTK (0.43) BTKFLT3PDE3BPDE3AGRM2
SCHEMBL12469271 0.78 NISCH (0.43) BTKGRM2
SCHEMBL12469700 0.77 BTK (0.40) BTKFLT3PDE3BPDE3AGRM5
SCHEMBL12469593 0.77 BTK (0.44) BTKPDE3BPDE3AGRM5GRM2
SCHEMBL12469863 0.76 BTK (0.42) BTKFLT3PDE3BPDE3AGRM2
SCHEMBL12469435 0.76 BTK (0.45) BTKFLT3PDE3BPDE3AGRM2
SCHEMBL12469516 0.76 GRM2 (0.40) BTKFLT3PDE3BPDE3AGRM5
SCHEMBL12469765 0.76 AURKA (0.40) BTKFLT3GRM5GRM2
SCHEMBL12469688 0.76 FLT3 (0.48) BTKFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed