SCHEMBL12469700

SCHEMBL12469700

Nc1ccc(-c2ccc(-c3nnc[nH]3)c3c2CNC3=O)c(F)c1.Nc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BTK Q06187 11/20 0.40
FLT3 P36888 1/20 0.36
GRM2 Q14416 1/20 0.33
KDR P35968 1/20 0.32
PIM1 P11309 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12469667 0.85 BTK (0.43) BTKFLT3GRM2PIM1PIM2
SCHEMBL12469435 0.82 BTK (0.45) BTKFLT3GRM2KDRPIM1
SCHEMBL12469532 0.82 BTK (0.42) BTKFLT3GRM2KDRPIM1
SCHEMBL12469863 0.80 BTK (0.42) BTKFLT3GRM2PIM1PIM2
SCHEMBL12469189 0.80 BTK (0.46) BTKFLT3KDRPIM1PIM2
SCHEMBL12469765 0.78 AURKA (0.40) BTKFLT3GRM2KDRGRM5
SCHEMBL12469688 0.78 FLT3 (0.48) BTKFLT3
Aniline SCHEMBL12469012 0.78 BTK (0.42) BTKFLT3KDRPIM1PIM2
SCHEMBL12469271 0.78 NISCH (0.43) BTKGRM2
SCHEMBL12469609 0.78 BTK (0.39) BTKFLT3GRM2KDRPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047017-A2 2,3-DIHYDRO-ISOINDOL-1-ONE DERIVATIVE AND A COMPOSITION COMPRISING THE SAME 크리스탈지노믹스(주) (KR) 2012-04-12 WO disclosed