SCHEMBL12474154

SCHEMBL12474154

CN1CCN([C@@H]2CCC[C@@H](CCC(N)=O)C2)CC1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 3/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
HIF1A Q16665 1/20 0.33
SIGMAR1 Q99720 3/20 0.33
L3MBTL3 Q96JM7 2/20 0.33
TP53 P04637 1/20 0.32
HSD11B1 P28845 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
BDKRB1 P46663 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6855190 0.74 NCF1 (0.48) ALDH1A1ATML3MBTL1HSD11B1HRH3
SCHEMBL23110427 0.73 SMN1; SMN2 (0.44) MEN1KMT2AALDH1A1ATML3MBTL1
SCHEMBL3594708 0.73 KDM4E (0.33) ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL30412623 0.73 GNAI3 (0.50) ALDH1A1ATML3MBTL1HSD11B1HRH3
SCHEMBL930589 0.72
SCHEMBL14098703 0.72 HPGD (0.37) MEN1KMT2AALDH1A1ATMHSD11B1
SCHEMBL1936961 0.71 TP53 (0.39) ALDH1A1ATML3MBTL1L3MBTL3TP53
SCHEMBL15986798 0.70 NCF1 (0.42) ALDH1A1L3MBTL1
SCHEMBL12474153 0.70 L3MBTL3 (0.36) L3MBTL1KDM4ESIGMAR1L3MBTL3TP53
SCHEMBL15088883 0.69 ALDH1A1 (0.53) ALDH1A1L3MBTL1KDM4EL3MBTL3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611810-A1 SUBSTITUTED TETRAHYDROPYRROLOPYRAZINE DERIVATIVES Grünenthal GmbH (DE) 2013-07-10 EP disclosed
WO-2012028331-A1 SUBSTITUTED TETRAHYDROPYRROLOPYRAZINE DERIVATIVES Grünenthal GmbH (DE) 2012-03-08 WO disclosed