SCHEMBL1247804

SCHEMBL1247804

CCOC(=O)N(c1ccccc1Cl)c1c(-c2ccc(CS(=O)(=O)c3ccc(CC(=O)O)cc3)cc2)noc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.37
NR1H4 Q96RI1 3/20 0.36
RORC P51449 2/20 0.36
PTGS2 P35354 1/20 0.36
NR4A2 P43354 1/20 0.36
GPBAR1 Q8TDU6 3/20 0.35
POLB P06746 2/20 0.35
MAPT P10636 2/20 0.35
ALDH1A1 P00352 3/20 0.34
PPARD Q03181 1/20 0.34
LPAR1 Q92633 1/20 0.34
LPAR2 Q9HBW0 1/20 0.34
LPAR3 Q9UBY5 1/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9902333 0.92 ALDH1A1 (0.35) NPSR1NR1H4GPBAR1POLBMAPT
SCHEMBL1245358 0.91 NR1H4 (0.42) NR1H4PTGS2GPBAR1POLBMAPT
SCHEMBL1245176 0.89 NR1H4 (0.40) NR1H4GPBAR1POLBMAPTALDH1A1
SCHEMBL1246186 0.89 PTGDR2 (0.38) NPSR1GPBAR1POLBMAPTALDH1A1
SCHEMBL1246477 0.88 NR1H4 (0.42) NR1H4GPBAR1MAPTALDH1A1PPARD
SCHEMBL3701141 0.87 LPAR1 (0.43) NPSR1NR1H4RORCMAPTALDH1A1
SCHEMBL1246467 0.86 NR1H4 (0.43) NR1H4PTGS2GPBAR1PPARDLPAR1
SCHEMBL1245335 0.85 NR1H4 (0.50) NR1H4MAPTPPARD
SCHEMBL1246476 0.85 NR1H4 (0.42) NR1H4GPBAR1MAPTALDH1A1PPARD
SCHEMBL1246346 0.84 SCN9A (0.38) NR1H4GPBAR1MAPTALDH1A1PPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed