SCHEMBL12482191

SCHEMBL12482191

O=NC(=O)c1ccnc(-c2cc(F)c(F)c(F)c2C2CCN(Cc3ccc(-c4ccc(F)cc4)cc3)CC2)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 2/20 0.40
KDM4A O75164 1/20 0.40
KDM5A P29375 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
GAA P10253 1/20 0.38
ACHE P22303 3/20 0.38
GSK3B P49841 3/20 0.38
BCHE P06276 1/20 0.38
AKT1 P31749 1/20 0.37
AKT2 P31751 1/20 0.37
HTR2A P28223 2/20 0.37
MCHR1 Q99705 2/20 0.37
CHRM4 P08173 1/20 0.37
SSTR5 P35346 1/20 0.37
CYP2D6 P10635 1/20 0.37
CHRM1 P11229 1/20 0.37
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1846809 0.90 PRKAA2 (0.42) KDM4CKDM4AKDM5AKDM5BGAA
SCHEMBL1847418 0.79 PRKAA2 (0.44) KDM4CKDM4AKDM5AKDM5BGAA
SCHEMBL1725767 0.75 GSK3B (0.45) ACHEGSK3BBCHEMCHR1
SCHEMBL1726693 0.75 MCHR1 (0.38) ACHEGSK3BBCHEHTR2AMCHR1
SCHEMBL1846811 0.74 MCHR1 (0.47) ACHEGSK3BBCHEHTR2AMCHR1
SCHEMBL12482193 0.74 OPRM1 (0.42) ACHEHTR2AMCHR1CHRM4CYP2D6
SCHEMBL12482196 0.73 MCHR1 (0.37) ACHEGSK3BBCHEHTR2AMCHR1
SCHEMBL1035443 0.68 AKT1 (0.41) KDM4CKDM4AKDM5AKDM5BAKT1
SCHEMBL1844021 0.67 WNK1 (0.43)
SCHEMBL1726547 0.66 GSK3B (0.48) ACHEGSK3BBCHEMCHR1CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012037282-A3 CATALYSTS AND METHODS FOR POLYMER SYNTHESIS NOVOMER, INC. (US) 2012-05-10 WO disclosed