SCHEMBL12489702

SCHEMBL12489702

Nc1nc2c(Cl)ncnc2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.36
ADORA3 P0DMS8 4/20 0.35
ALDH1A1 P00352 2/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.35
MAPK3 P27361 1/20 0.35
XDH P47989 1/20 0.35
HBB P68871 1/20 0.35
PAX8 Q06710 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
PMP22 Q01453 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MMP12 P39900 2/20 0.34
NUDT1 P36639 1/20 0.34
PNP P00491 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016628 0.81 CHEK1 (0.37) CHEK1ADORA3ALDH1A1KDM4EAURKA
SCHEMBL11125305 0.79 ALDH1A1 (0.35) ADORA3ALDH1A1USP2TP53HPGD
SCHEMBL42313 0.78 ADORA2A (0.42) ADORA3ALDH1A1USP2TP53HPGD
SCHEMBL17289600 0.78 ADORA2A (0.43) CHEK1ADORA3AURKAADORA2AADORA1
SCHEMBL9544738 0.78 ADORA3 (0.40) CHEK1ADORA3KDM4EAURKAHTT
SCHEMBL6831168 0.75 CSNK2A2 (0.41) ADORA3ALDH1A1USP2TP53HPGD
SCHEMBL6829678 0.75 ALDH1A1 (0.35) ADORA3ALDH1A1USP2TP53HPGD
SCHEMBL6826186 0.75 ALDH1A1 (0.35) ADORA3ALDH1A1USP2TP53HPGD
SCHEMBL28995610 0.75 MMP12 (0.36) ADORA3ALDH1A1USP2TP53HPGD
SCHEMBL1868817 0.73 ADORA2A (0.43) ALDH1A1HPGDLMNAKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7972994-B2 Methods for synthesis of encoded libraries GLAXOSMITHKLINE LLC (US) 2011-07-05 US disclosed
US-20070042401-A1 Methods for synthesis of encoded libraries PRAECIS PHARMACEUTICALS, INC. (US) 2007-02-22 US disclosed