SCHEMBL124935

SCHEMBL124935

CCc1ccccc1C(=CCCN)c1ccccc1C

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 12/20 0.40
TAAR1 Q96RJ0 1/20 0.40
HPGD P15428 2/20 0.39
SHBG P04278 1/20 0.38
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GPR52 Q9Y2T5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724891 0.89 SLC6A1 (0.43) SLC6A1TAAR1HPGDGPR52
SCHEMBL6546899 0.80 HPGD (0.45) HPGDSHBGKDM4EALDH1A1GPR52
SCHEMBL5724863 0.72 SLC6A1 (0.43) SLC6A1HPGDGPR52
SCHEMBL5402022 0.70 HPGD (0.51) HPGDSHBGKDM4EALDH1A1
SCHEMBL6546961 0.70 HPGD (0.47) HPGDSHBGKDM4EALDH1A1
SCHEMBL1318497 0.68 SLC6A1 (0.40) SLC6A1GPR52
SCHEMBL7923183 0.68 ERCC5 (0.39) SLC6A1HPGDGPR52
SCHEMBL11348407 0.67 SHBG (0.67) HPGDSHBGKDM4EALDH1A1
SCHEMBL14415792 0.67 MAOA (0.42) SLC6A1HPGDALDH1A1
SCHEMBL19012291 0.66 TAAR1 (0.41) TAAR1HPGDKDM4EALDH1A1GPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2446903-A2 Methods, compositions, and kits for treating pain and pruritis President and Fellows of Harvard College (US) 2012-05-02 EP disclosed
EP-2425858-A2 Compositions for treating pain and pruritus President and Fellows of Harvard College (US) 2012-03-07 EP disclosed