SCHEMBL1249526

SCHEMBL1249526

CS(=O)(=O)N(F)[C@@](F)(CCCN)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ODC1 P11926 2/20 0.40
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
BLM P54132 1/20 0.38
PMP22 Q01453 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA9 Q16790 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7940896 0.79 ODC1 (0.44) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL29001334 0.77 ODC1 (0.43) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL30116554 0.74 ODC1 (0.50) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL6151309 0.73 ODC1 (0.41) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL6151308 0.73 ODC1 (0.41) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL5069038 0.72 CHRM2 (0.40) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL1249523 0.71 ODC1 (0.41) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL28113559 0.65 ODC1 (0.54) ODC1KDM4ELMNAMAPTRAB9A
Trifluoroacetic Acid SCHEMBL31080805 0.65 ODC1 (0.48) ODC1KDM4ELMNAMAPTRAB9A
SCHEMBL15909004 0.63 CES2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678305-A2 PROTOZOAN STRAINS OF REDUCED VIRULENCE AND USE THEREOF Institut de Recherche pour le Développement ( IRD) (FR) 2006-07-12 EP claimed
WO-2005044844-A2 PROTOZOAN STRAINS OF REDUCED VIRULENCE AND USE THEREOF INSTITUT DE RECHERCHE POUR LE DEVELOPPEMENT (FR) 2005-05-19 WO claimed
EP-3554531-A1 TREATMENT OF AGE-RELATED DEGENERATION AND OTHER EYE DISEASES WITH APOLIPOPROTEIN MIMETICS MacRegen, Inc. (US) 2019-10-23 EP disclosed
WO-2018139991-A1 TREATMENT OF AGE-RELATED DEGENERATION AND OTHER EYE DISEASES WITH APOLIPOPROTEIN MIMETICS MACREGEN, INC. (US) 2018-08-02 WO disclosed
EP-3204379-A1 PYRROLIDINE AMIDE COMPOUNDS AS HISTONE DEMETHYLASE INHIBITORS Genentech, Inc. (US) 2017-08-16 EP disclosed
WO-2016057924-A1 PYRROLIDINE AMIDE COMPOUNDS AS HISTONE DEMETHYLASE INHIBITORS GENENTECH, INC. (US) 2016-04-14 WO disclosed
WO-2013075120-A1 METHODS OF TREATING CANCER WITH HERBACETIN REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2013-05-23 WO disclosed
EP-2278969-A2 INHIBITORS OF JANUS KINASES Merck Sharp & Dohme Corp. (US) 2011-02-02 EP disclosed
WO-2010011375-A2 INHIBITORS OF JANUS KINASES MERCK & CO., INC. (US) 2010-01-28 WO disclosed
WO-2005116050-A1 STEROID-HORMONE CONJUGATES WITH POLYAMINES AND THEIR THERAPEUTIC USE AS ANTI-CANCER AND ANGIOSTATIC AGENTS HUNTER-FLEMING LIMITED (GB) 2005-12-08 WO disclosed