SCHEMBL29147689

SCHEMBL29147689

CC1CCCC(C)N1Cc1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
LTA4H P09960 1/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ACHE P22303 3/20 0.40
HRH3 Q9Y5N1 2/20 0.40
BCHE P06276 1/20 0.39
BACE1 P56817 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CHEK1 O14757 1/20 0.39
KCNH2 Q12809 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1427504 1.00 ALDH1A1 (0.42) ALDH1A1LTA4HKDM4EHPGDTDP1
SCHEMBL16215682 0.83 ALDH1A1 (0.52) ALDH1A1LTA4HL3MBTL1ACHEHRH3
SCHEMBL17533290 0.83 ALDH1A1 (0.44) ALDH1A1LTA4HKDM4EACHEHRH3
SCHEMBL13405849 0.83 ALDH1A1 (0.50) ALDH1A1LTA4HKDM4EHPGDACHE
SCHEMBL3146950 0.81 ALDH1A1 (0.63) ALDH1A1LTA4HKDM4ETDP1ACHE
SCHEMBL17055247 0.81 LTA4H (0.54) ALDH1A1LTA4HKDM4EHPGDACHE
SCHEMBL18557 0.81 LTA4H (0.54) ALDH1A1LTA4HKDM4EHPGDACHE
SCHEMBL12499953 0.80 KDM4E (0.40) ALDH1A1KDM4EL3MBTL1ACHEHRH3
SCHEMBL12499770 0.80 ALDH1A1 (0.40) ALDH1A1KDM4EHPGDSIGMAR1POLB
SCHEMBL12463216 0.80 OPRK1 (0.45) ALDH1A1L3MBTL1SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116964046-B PLK4 inhibitors and uses thereof 上海齐鲁制药研究中心有限公司 2024-04-19 CN disclosed
CN-116964046-A PLK4 inhibitors and uses thereof 上海齐鲁制药研究中心有限公司 2023-10-27 CN disclosed
WO-2022184049-A1 PLK4 INHIBITOR AND USE THEREOF 上海齐鲁制药研究中心有限公司 2022-09-09 WO disclosed