SCHEMBL12628172

SCHEMBL12628172

O=C(NS(=O)(=O)c1ccccc1)[C@@H]1CC[C@H](c2ccccc2)N(S(=O)(=O)c2ccccc2)C1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
RAB9A P51151 2/20 0.57
KMT2A Q03164 1/20 0.57
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43
APH1A Q96BI3 1/20 0.43
PSENEN Q9NZ42 1/20 0.43
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPC1 O15118 1/20 0.40
MMP2 P08253 2/20 0.40
MMP9 P14780 2/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
EPHX2 P34913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014926 1.00 ALDH1A1 (0.57) ALDH1A1RAB9AKMT2APSEN1PSEN2
SCHEMBL12629087 0.85 ALDH1A1 (0.65) ALDH1A1RAB9AKMT2APSEN1PSEN2
SCHEMBL2011747 0.85 ALDH1A1 (0.65) ALDH1A1RAB9AKMT2APSEN1PSEN2
SCHEMBL2013828 0.85 ALDH1A1 (0.57) ALDH1A1RAB9AKMT2ANPC1
SCHEMBL12629075 0.85 ALDH1A1 (0.57) ALDH1A1RAB9AKMT2ANPC1
SCHEMBL12628511 0.82 ALDH1A1 (0.53) ALDH1A1RAB9AKMT2APSEN1PSEN2
SCHEMBL2010855 0.82 ALDH1A1 (0.53) ALDH1A1RAB9AKMT2APSEN1PSEN2
SCHEMBL12628159 0.82 ALDH1A1 (0.54) ALDH1A1RAB9AKMT2A
SCHEMBL2018212 0.82 ALDH1A1 (0.53) ALDH1A1RAB9AKMT2APSEN1PSEN2
SCHEMBL12628187 0.82 ALDH1A1 (0.53) ALDH1A1RAB9AKMT2APSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO disclosed