SCHEMBL1272033

SCHEMBL1272033

C=C(SCCCCC)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CES2 O00748 3/20 0.43
CES1 P23141 3/20 0.43
PTGS2 P35354 4/20 0.42
NAAA Q02083 1/20 0.41
ESR1 P03372 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19391886 0.94 ALDH1A1 (0.49) ALDH1A1NPSR1CES2CES1PTGS2
SCHEMBL12900930 0.88 ALDH1A1 (0.41) ALDH1A1NPSR1CES2CES1PTGS2
SCHEMBL12900928 0.88 CES2 (0.44) ALDH1A1NPSR1CES2CES1PTGS2
SCHEMBL23837678 0.86 CES2 (0.38) ALDH1A1NPSR1CES2CES1PTGS2
SCHEMBL1270960 0.80 LMNA (0.49) ALDH1A1POLB
SCHEMBL19391813 0.79 SMN1; SMN2 (0.37) ALDH1A1NPSR1
SCHEMBL19677301 0.78 HDAC3 (0.46) ALDH1A1NPSR1CES2CES1
SCHEMBL6057406 0.78 CES2 (0.51) ALDH1A1NPSR1CES2CES1PTGS2
SCHEMBL12900922 0.76 ALDH1A1 (0.42) ALDH1A1NPSR1CES2CES1PTGS2
SCHEMBL10797615 0.76 CES2 (0.53) ALDH1A1NPSR1CES2CES1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140142319-A1 ORGANOACTINIDE-, ORGANOLANTHANIDE-, AND ORGANOGROUP-4-MEDIATED HYDROTHIOLATION OF TERMINAL ALKYNES WITH ALIPHATIC, AROMATIC AND BENZYLIC THIOLS NORTHWESTERN UNIVERSITY (US) 2014-05-22 US claimed
US-20110040098-A1 Organoactinide-, Organolanthanide-, and OrganoGroup-4-Mediated Hydrothiolation of Terminal Alkynes with Aliphatic, Aromatic and Benzylic Thiols NATIONAL SCIENCE FOUNDATION 2011-02-17 US claimed
US-20140142319-A1 ORGANOACTINIDE-, ORGANOLANTHANIDE-, AND ORGANOGROUP-4-MEDIATED HYDROTHIOLATION OF TERMINAL ALKYNES WITH ALIPHATIC, AROMATIC AND BENZYLIC THIOLS NORTHWESTERN UNIVERSITY (US) 2014-05-22 US disclosed
US-20140142319-A1 ORGANOACTINIDE-, ORGANOLANTHANIDE-, AND ORGANOGROUP-4-MEDIATED HYDROTHIOLATION OF TERMINAL ALKYNES WITH ALIPHATIC, AROMATIC AND BENZYLIC THIOLS NORTHWESTERN UNIVERSITY (US) 2014-05-22 US disclosed
US-20140142319-A1 ORGANOACTINIDE-, ORGANOLANTHANIDE-, AND ORGANOGROUP-4-MEDIATED HYDROTHIOLATION OF TERMINAL ALKYNES WITH ALIPHATIC, AROMATIC AND BENZYLIC THIOLS NORTHWESTERN UNIVERSITY (US) 2014-05-22 US disclosed
US-8609902-B2 Organoactinide-, organolanthanide-, and organogroup-4-mediated hydrothiolation of terminal alkynes with aliphatic, aromatic and benzylic thiols NORTHWESTERN UNIVERSITY (US) 2013-12-17 US disclosed
US-20110040098-A1 Organoactinide-, Organolanthanide-, and OrganoGroup-4-Mediated Hydrothiolation of Terminal Alkynes with Aliphatic, Aromatic and Benzylic Thiols NATIONAL SCIENCE FOUNDATION 2011-02-17 US disclosed
US-20110040098-A1 Organoactinide-, Organolanthanide-, and OrganoGroup-4-Mediated Hydrothiolation of Terminal Alkynes with Aliphatic, Aromatic and Benzylic Thiols NATIONAL SCIENCE FOUNDATION 2011-02-17 US disclosed
US-20110040098-A1 Organoactinide-, Organolanthanide-, and OrganoGroup-4-Mediated Hydrothiolation of Terminal Alkynes with Aliphatic, Aromatic and Benzylic Thiols NATIONAL SCIENCE FOUNDATION 2011-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140142319-A1 ORGANOACTINIDE-, ORGANOLANTHANIDE-, AND ORGANOGROUP-4-MEDIATED HYDROTHIOLATION OF TERMINAL ALKYNES WITH ALIPHATIC, AROMATIC AND BENZYLIC THIOLS OR10J3, HCN4, HVCN1 ALDH1A1 283/4885NPSR1 3210/4885CES2 1994/4885
US-20110040098-A1 Organoactinide-, Organolanthanide-, and OrganoGroup-4-Mediated Hydrothiolation of Terminal Alkynes with Aliphatic, Aromatic and Benzylic Thiols OR10J3, HCN4, HVCN1 ALDH1A1 283/4885NPSR1 3210/4885CES2 1994/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.