SCHEMBL1274871

SCHEMBL1274871

O=C(O)C(Cc1ccccc1)n1c(-c2ccccc2)c(Cl)nc(Cl)c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
HSD17B10 Q99714 2/20 0.49
MAPT P10636 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
MEN1 O00255 2/20 0.49
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
PTPN7 P35236 1/20 0.49
RECQL P46063 1/20 0.49
BLM P54132 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
AADAT Q8N5Z0 1/20 0.47
ALDH1A1 P00352 3/20 0.45
PKM P14618 1/20 0.45
GAA P10253 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44
HDAC8 Q9BY41 3/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1274295 0.87 HSD17B10 (0.47) KMT2AHSD17B10MAPTL3MBTL1MEN1
SCHEMBL7453183 0.83 F7 (0.51)
SCHEMBL7019887 0.83 KMT2A (0.57) KMT2AHSD17B10MAPTL3MBTL1MEN1
SCHEMBL5791501 0.75 POLB (0.69) KMT2AHSD17B10MAPTL3MBTL1MEN1
SCHEMBL2454105 0.75 POLB (0.69) KMT2AHSD17B10MAPTL3MBTL1MEN1
SCHEMBL6989591 0.72 ALDH1A1 (0.34) KMT2AHSD17B10MAPTMEN1KDM4E
SCHEMBL3594973 0.70 KDM4E (0.49) HSD17B10KDM4E
SCHEMBL1746215 0.69 MAPT (0.59) KMT2AHSD17B10MAPTL3MBTL1MEN1
SCHEMBL9194175 0.67 KMT2A (0.75) KMT2AHSD17B10MAPTL3MBTL1MEN1
SCHEMBL9554515 0.67 MAPT (1.00) KMT2AHSD17B10MAPTL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7893079-B2 Substituted monocyclic CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2011-02-22 US disclosed