SCHEMBL12825633

SCHEMBL12825633

O=C(O)c1cn(C2CC2)c2c3c(c(F)cc2c1=O)N1CCNCC1CCO3

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
KDM4E B2RXH2 6/20 0.50
HPGD P15428 5/20 0.50
HSD17B10 Q99714 5/20 0.50
TOP2A P11388 4/20 0.50
TOP2B Q02880 4/20 0.50
AADAT Q8N5Z0 2/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
KCNH2 Q12809 5/20 0.49
POLB P06746 3/20 0.49
OPRM1 P35372 2/20 0.49
PRKD3 O94806 1/20 0.49
ALOX15 P16050 1/20 0.49
CLK2 P49760 1/20 0.49
CLK4 Q9HAZ1 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12836940 1.00 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL12825615 0.88 ADRB2 (0.48) ALDH1A1KDM4EHPGDHSD17B10AADAT
SCHEMBL115248 0.87 AADAT (0.53) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL12825263 0.85 AADAT (0.54) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL12819590 0.84 LMNA (0.54) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL12825636 0.82 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL12819586 0.82 TOP2A (0.52) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL117484 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL116011 0.81 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL116382 0.81 AADAT (0.58) ALDH1A1KDM4EHPGDHSD17B10TOP2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011031740-A1 ANTIBACTERIAL FLUOROQUINOLONE ANALOGS ACHAOGEN, INC. (US) 2011-03-17 WO disclosed