SCHEMBL12835629

SCHEMBL12835629

O=C(O)Cc1cccc2c(=O)cc(-c3ccc(-c4ccccc4)c(-c4ccccc4)c3)oc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.53
CYP1A2 P05177 6/20 0.52
CYP3A4 P08684 4/20 0.52
CYP2C19 P33261 3/20 0.52
STAT6 P42226 1/20 0.52
CYSLTR1 Q9Y271 1/20 0.46
CYP1A1 P04798 6/20 0.46
CYP1B1 Q16678 6/20 0.46
CYP19A1 P11511 4/20 0.45
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 3/20 0.45
TP53 P04637 3/20 0.45
MAPT P10636 3/20 0.45
HPGD P15428 3/20 0.45
MAPK1 P28482 3/20 0.45
HSD17B10 Q99714 3/20 0.45
PRKDC P78527 2/20 0.45
CYP2C9 P11712 2/20 0.45
PDE5A O76074 1/20 0.45
ABCB1 P08183 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12835503 0.89 CYP1A2 (0.60) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
Mitoflaxone SCHEMBL106705 0.89 CYP1A2 (0.62) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL12835325 0.86 CDK1 (0.48) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL12835292 0.84 CYP2D6 (0.51) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL7083117 0.83 CYP1A2 (0.59) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9328614 0.83 CYP1A2 (0.59) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL12835531 0.83 CYP1A2 (0.54) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL7083153 0.83 CYP2D6 (0.54) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL12835338 0.83 TDP1 (0.57) CYP2D6CYP1A2CYP3A4CYP2C19STAT6
SCHEMBL9327546 0.82 CYP1A2 (0.58) CYP2D6CYP1A2CYP3A4CYP2C19STAT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011023287-A1 USE OF FAA AND ITS DERIVATIVES IN COSMETICS AND DERMATOLOGY MERCK PATENT GMBH (DE) 2011-03-03 WO disclosed