SCHEMBL12836282

SCHEMBL12836282

COc1ccccc1C1(O)CC2CCCNC2C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.51
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
HSD11B1 P28845 1/20 0.41
HTR1A P08908 3/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM5 P08912 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39
ADRA1A P35348 2/20 0.38
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12836645 0.80 OPRM1 (0.36) SIGMAR1DRD2DRD3OPRM1OPRL1
SCHEMBL12836222 0.76 OPRM1 (0.41) SIGMAR1OPRM1OPRD1OPRK1OPRL1
SCHEMBL6747981 0.74 SIGMAR1 (0.56) SIGMAR1DRD2DRD3ALDH1A1TSHR
SCHEMBL12179327 0.71 CHRM2 (0.38) SIGMAR1HSD11B1HTR1ACHRM2CHRM4
SCHEMBL17376311 0.71 SIGMAR1 (0.43) SIGMAR1DRD2DRD3CHRNB4CHRNA3
SCHEMBL8586983 0.70 SLC6A4 (0.61) SIGMAR1DRD2DRD3ALDH1A1TSHR
SCHEMBL7542807 0.69 SIGMAR1 (0.72) SIGMAR1DRD2DRD3ALDH1A1TSHR
SCHEMBL29965651 0.69 SIGMAR1 (0.72) SIGMAR1DRD2DRD3ALDH1A1TSHR
SCHEMBL12836642 0.69 HTR1A (0.50) SIGMAR1DRD2DRD3HTR1ACHRM2
SCHEMBL30368868 0.68 SIGMAR1 (1.00) SIGMAR1DRD2DRD3CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011033255-A1 (4-PHENYL-PIPERIDIN-1-YL)-[5-1H-PYRAZOL-4YL)-THIOPHEN-3-YL]-METHANONE COMPOUNDS AND THEIR USE THE UNIVERSITY OF EDINBURGH (GB) 2011-03-24 WO disclosed