SCHEMBL128398

SCHEMBL128398

[CH2]c1ccc(C(O)(C(F)(F)F)C(F)(F)F)cc1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 15/20 0.56
NR1H3 Q13133 15/20 0.56
MLYCD O95822 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL131990 0.87 NR1H2 (0.68) NR1H2NR1H3MLYCDSMN1; SMN2
Water SCHEMBL1684070 0.84 NR1H2 (0.65) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL130132 0.79 NR1H2 (0.52) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL24901413 0.79 NR1H2 (0.61) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL9621271 0.79 NR1H2 (0.60) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL6808538 0.77 ESR1 (0.61) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL8021367 0.77 NR1H2 (0.58) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL1516045 0.77 ESR1 (0.61) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL17054 0.75 NR1H2 (0.56) NR1H2NR1H3MLYCDSMN1; SMN2
SCHEMBL14593303 0.75 NR1H2 (0.61) NR1H2NR1H3MLYCDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102026986-B Hexafluoroisopropanol derivatives MERCK SHARP & DOHME B.V. (NL) 2014-10-29 CN disclosed
US-8450319-B2 Pyrrolopyridazinone compound UBE INDUSTRIES, LTD. (JP) 2013-05-28 US disclosed
EP-1982986-B1 PYRROLOPYRIDAZINONE COMPOUND AS PDE4 INHIBITOR UBE INDUSTRIES (JP) 2012-03-07 EP disclosed
CN-101374844-A Pyrrolopyridazinone compound UBE INDUSTRIES (JP) 2009-02-25 CN disclosed
US-20090036453-A1 Pyrrolopyridazinone Compound UBE INDUSTRIES, LTD. (JP) 2009-02-05 US disclosed
EP-1982986-A1 PYRROLOPYRIDAZINONE COMPOUND Ube Industries, Ltd. (JP) 2008-10-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090036453-A1 Pyrrolopyridazinone Compound CBR3, CBR1, CYC1 NR1H2 857/4885NR1H3 1338/4885MLYCD 481/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.