SCHEMBL10069601

SCHEMBL10069601

CC(C)c1c(-c2ccc(F)cc2)n(COCc2ccccc2)c(=O)n(O)c1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
GRM5 P41594 1/20 0.34
CYP1A2 P05177 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HMGCR P04035 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ASAH1 Q13510 1/20 0.34
ELANE P08246 1/20 0.34
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP3A4 P08684 2/20 0.33
HPGD P15428 1/20 0.33
GNRHR P30968 1/20 0.33
ERCC5 P28715 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10069611 0.96 L3MBTL1 (0.36) ALDH1A1L3MBTL1GRM5CYP1A2HMGCR
SCHEMBL10069619 0.95 KDM5B (0.34) L3MBTL1CYP3A4GNRHR
SCHEMBL10069590 0.92 ALDH1A1 (0.39) ALDH1A1ELANEERCC5FEN1MAPK1
SCHEMBL10069602 0.90 ALDH1A1 (0.39) ALDH1A1L3MBTL1MEN1KMT2AKDM4E
SCHEMBL10069596 0.90 MAPT (0.36) ALDH1A1CYP1A2CASP1CASP7HSD17B10
SCHEMBL10069594 0.89 MAPT (0.38) ALDH1A1GRM5CYP1A2HSD17B10KDM4E
SCHEMBL10069592 0.87 MEN1 (0.40) ALDH1A1MEN1KMT2AKDM4EELANE
SCHEMBL10069591 0.86 ESR1 (0.35) ALDH1A1CYP1A2MEN1KMT2AERCC5
SCHEMBL10069598 0.85 TP53 (0.33) GRM5HMGCR
SCHEMBL10069595 0.85 ALDH1A1 (0.38) ALDH1A1GRM5ERCC5FEN1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed