SCHEMBL12880577

SCHEMBL12880577

BrC(c1ccccc1)c1ccc(C(Br)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
TRPA1 O75762 1/20 0.48
DPP4 P27487 2/20 0.45
F2 P00734 1/20 0.45
TSHR P16473 1/20 0.45
HTR2A P28223 2/20 0.42
TAAR1 Q96RJ0 2/20 0.41
CYP2D6 P10635 1/20 0.39
SRC P12931 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
LMNA P02545 2/20 0.38
HRH1 P35367 1/20 0.38
MTOR P42345 1/20 0.38
RAB9A P51151 1/20 0.38
GRM7 Q14831 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL67123 0.97 CES2 (0.50) CES2CES1TRPA1DPP4F2
SCHEMBL12880591 0.91 CHRNB2 (0.50) CES2CES1TRPA1DPP4F2
SCHEMBL8721667 0.89 CHRNB2 (0.54) CES2CES1TRPA1HTR2ATAAR1
SCHEMBL11576225 0.89 HTR2A (0.58) CES2CES1TRPA1HTR2ALMNA
SCHEMBL7520122 0.87 LMNA (0.42) CES2CES1TRPA1LMNA
SCHEMBL10766035 0.87 CES2 (0.39) CES2CES1TRPA1DPP4F2
SCHEMBL14528562 0.87 CES2 (0.39) CES2CES1TRPA1DPP4F2
SCHEMBL1528588 0.87 IDO1 (0.54) TRPA1TSHRCYP2D6LMNAMAPK1
SCHEMBL1272990 0.87 LMNA (0.48) CES2CES1TRPA1TSHRLMNA
SCHEMBL30961545 0.87 PDPK1 (0.42) CES2CES1TRPA1DPP4F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884175-B2 polymerizing one or more monomers containing dihalogen containing substituted biaryls, via a base-induced dehydrohalogenation MERCK PATENT GMBH (DE) 2011-02-08 US disclosed
US-7884175-B2 polymerizing one or more monomers containing dihalogen containing substituted biaryls, via a base-induced dehydrohalogenation MERCK PATENT GMBH (DE) 2011-02-08 US disclosed
EP-1623471-B1 METHOD FOR CONTROLLING THE MOLECULAR WEIGHT DURING POLY(ARYLENE VINYLENE) SYNTHESIS, AND POLYMERS PRODUCED THEREWITH MERCK PATENT GMBH (DE) 2007-05-30 EP disclosed